Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A673 CCLE 1.357 25.9 25.9 0.000 0
HOS CCLE 3.913 N/A 0.127 92.175 0
MG-63 CCLE 0.693 15.3 10 40.000 0
MHH-ES-1 CCLE 9.366 8.09 8.09 0.000 0
Saos-2 CCLE 0.540 12.1 12.1 0.000 0
SJSA-1 CCLE 4.631 116 116 0.000 0
SK-ES-1 CCLE 6.852 N/A 2.43 53.599 0.0514
SW 1353 CCLE 2.773 370 370 0.000 0
TC-71 CCLE 1.113 N/A 0.0132 97.775 0
U-2-OS CCLE 5.060 36.1 36.1 0.000 0
ES8 GDSC1000 7.895 N/A 1e+06 84.210 0
EW-18 GDSC1000 1.519 N/A 0.101 96.962 0
SK-PN-DW GDSC1000 5.172 121 121 0.000 0
EW-11 GDSC1000 9.066 N/A 0.0702 84.988 0.0288
SK-ES-1 GDSC1000 3.266 N/A 0.933 77.090 0.011
TC-71 GDSC1000 0.153 4.64 4.64 0.000 0
ES7 GDSC1000 2.744 N/A 1e+06 94.512 0
ES4 GDSC1000 19.684 N/A 0.0257 74.791 0.118
SK-NEP-1 GDSC1000 1.198 N/A 1.77 72.326 0.00185
NOS-1 GDSC1000 23.296 13.3 13.3 0.000 0
ES6 GDSC1000 28.592 N/A 2.31e-06 71.408 0.207
EW-1 GDSC1000 0.885 N/A 1.02 92.836 0
SJSA-1 GDSC1000 4.821 N/A 2.69e+03 90.358 0
EW-24 GDSC1000 36.907 0.317 0.0338 49.612 0.307
ES3 GDSC1000 0.354 N/A 0.116 99.311 0
ES5 GDSC1000 0.000 N/A 0.00781 100.000 0
EW-13 GDSC1000 0.000 N/A 0.00781 100.000 0
VA-ES-BJ GDSC1000 2.380 N/A 0.0291 96.878 0
EW-12 GDSC1000 0.000 N/A 0.00781 100.000 0
ES1 GDSC1000 42.395 N/A 1e-06 57.605 0.36
EW-16 GDSC1000 3.553 2.45 2.45 0.000 0
EW-3 GDSC1000 0.000 N/A 0.00781 100.000 0
A673 gCSI 3.906 522 522 0.000 0
MHH-ES-1 gCSI 1.267 178 178 0.000 0
TC-71 gCSI 7.618 39.7 39.7 0.000 0
U-2-OS gCSI 13.489 N/A 0.475 65.316 0.0581
SW 1353 CTRPv2 3.379 N/A 12.5 78.904 0.0157
U-2-OS CTRPv2 8.805 55.1 24.4 28.711 0.0577
MHH-ES-1 CTRPv2 8.950 N/A 9.16 52.974 0.0669
SJSA-1 CTRPv2 1.911 N/A 29.3 75.782 0.00818
SK-N-MC CTRPv2 9.427 N/A 5.76 59.770 0.0727
HOS CTRPv2 6.475 1.28e+03 1.28e+03 0.000 0
A673 CTRPv2 6.914 N/A 6.77 68.418 0.0472
MG-63 CTRPv2 3.731 N/A 38.7 61.162 0.012
TC-71 CTRPv2 5.501 N/A 13.2 64.559 0.0346
G-292;clone A141B1 CTRPv2 7.391 484 484 0.000 0
SK-ES-1 CTRPv2 16.319 7.79 3.82 40.426 0.138
Hs 888.T CTRPv2 21.629 8.86 3.03 29.091 0.17
Saos-2 CTRPv2 4.799 37.5 37.5 0.000 0
Hs 822.T CTRPv2 4.185 N/A 5.72 82.196 0.0171
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