Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MMAC-SF GDSC1000 40.584 0.11 0.11 0.000 0.363
A375 GDSC1000 77.282 0.0117 0.0116 1.020 0.748
WM902B GDSC1000 16.295 0.496 0.496 0.000 0.125
CP50-MEL-B GDSC1000 8.775 N/A 0.162 73.594 0.051
A431 GDSC1000 66.617 0.0218 0.0206 3.601 0.629
CHL-1 GDSC1000 61.673 0.031 0.031 0.000 0.574
WM278 GDSC1000 29.563 0.235 0.235 0.000 0.24
K4 GDSC1000 82.106 0.0099 0.00981 0.949 0.801
WM-115 GDSC1000 9.282 N/A 0.0117 81.435 0
SK-MEL-3 GDSC1000 37.307 0.139 0.139 0.000 0.32
WM35 GDSC1000 37.070 0.14 0.14 0.000 0.319
WM793B GDSC1000 68.330 0.00471 0.00471 0.000 0.648
MKL-1-subclone-2 GDSC1000 50.112 0.061 0.0598 2.179 0.471
DJM-1 GDSC1000 42.858 0.0872 0.0678 12.621 0.373
COLO-783 GDSC1000 11.231 20.8 20.8 0.000 0
C32 GDSC1000 7.326 N/A 0.00198 85.349 0
COLO-679 GDSC1000 69.829 0.0146 0.0128 10.161 0.665
MCC13 GDSC1000 8.535 N/A 0.362 55.909 0.0543
SK-MEL-2 GDSC1000 26.951 0.239 0.239 0.000 0.234
G-MEL GDSC1000 55.446 0.0417 0.0373 4.897 0.505
CP66-MEL GDSC1000 6.303 1.22 1.22 0.000 0
GAK GDSC1000 32.205 0.206 0.206 0.000 0.262
MKL-2 GDSC1000 56.876 0.0429 0.0426 0.472 0.53
WM1158 GDSC1000 52.469 0.0518 0.0504 3.352 0.498
G-361 GDSC1000 64.177 0.0231 0.0231 0.000 0.602
UISO-MCC-1 GDSC1000 47.587 0.0777 0.0777 0.000 0.418
WM239A GDSC1000 9.634 0.619 0.619 0.000 0.0807
MEL-JUSO GDSC1000 69.615 0.0132 0.0132 0.000 0.662
HMV-II GDSC1000 70.899 0.00843 0.00843 0.000 0.677
K19 GDSC1000 26.962 0.304 0.304 0.000 0.209
IPC-298 GDSC1000 37.319 0.155 0.155 0.000 0.309
HT-144 GDSC1000 76.312 0.00275 0.00275 0.000 0.737
A253 GDSC1000 56.578 0.0368 0.0318 8.442 0.519
A2058 GDSC1000 69.200 0.0198 0.0196 0.664 0.658
MZ2-MEL GDSC1000 61.929 0.0281 0.0281 0.000 0.577
451Lu GDSC1000 39.496 0.122 0.122 0.000 0.341
A388 GDSC1000 59.931 0.028 0.0228 8.651 0.555
RPMI-7951 GDSC1000 38.119 0.128 0.128 0.000 0.336
SK-MEL-24 GDSC1000 17.655 0.915 0.915 0.000 0.11
MZ7-mel GDSC1000 40.761 0.111 0.111 0.000 0.358
Mewo GDSC1000 7.969 2.51 2.51 0.000 0
COLO-792 GDSC1000 20.893 31.1 31.1 0.000 0
RVH-421 GDSC1000 38.284 0.177 0.177 0.000 0.314
SK-MEL-1 GDSC1000 1.734 1.29 1.29 0.000 0
SH-4 GDSC1000 46.509 0.0816 0.0778 1.682 0.406
IST-MEL1 GDSC1000 60.618 0.0163 0.0123 23.420 0.564
IGR-37 GDSC1000 52.175 0.0563 0.0563 0.000 0.475
Hs 940.T GDSC1000 49.098 0.0695 0.0695 0.000 0.434
MCC26 GDSC1000 8.408 0.928 0.928 0.000 0.0525
VMRC-MELG GDSC1000 9.032 0.654 0.654 0.000 0.0731
IGR-1 GDSC1000 55.838 0.0405 0.0366 6.214 0.513
WM1552C GDSC1000 53.149 0.0485 0.0485 0.000 0.479
LB2518-MEL GDSC1000 23.970 0.377 0.377 0.000 0.181
Hs 939.T GDSC1000 31.552 0.203 0.203 0.000 0.261
A101D GDSC1000 55.810 0.0426 0.0426 0.000 0.509
SK-MEL-30 GDSC1000 59.183 0.0346 0.0336 1.431 0.546
LB373-MEL-D GDSC1000 40.654 0.156 0.156 0.000 0.341
COLO-800 GDSC1000 44.242 0.0887 0.0887 0.000 0.404
K8 GDSC1000 16.032 0.433 0.433 0.000 0.138
COLO-829 GDSC1000 15.608 2.29 0.267 44.372 0.0963
A2058 gCSI 71.060 0.0362 0.0357 1.015 0.683
A375 gCSI 68.189 0.047 0.0464 0.766 0.651
A431 gCSI 48.332 0.287 0.287 0.000 0.445
C32 gCSI 38.725 0.378 0.295 19.326 0.358
CHL-1 gCSI 56.439 0.139 0.139 0.000 0.527
COLO-679 gCSI 51.635 0.214 0.214 0.000 0.48
COLO-800 gCSI 50.766 0.229 0.227 0.366 0.471
COLO-829 gCSI 49.081 0.269 0.269 0.000 0.451
G-361 gCSI 51.199 0.222 0.222 0.000 0.479
HMV-II gCSI 27.974 1 0.704 26.562 0.251
Hs 294T gCSI 60.024 0.0966 0.0966 0.000 0.558
Hs 695T gCSI 38.133 0.244 0.166 30.040 0.348
Hs 852.T gCSI 33.283 0.811 0.739 11.319 0.314
IGR-1 gCSI 49.415 0.26 0.26 0.000 0.459
IGR-37 gCSI 47.630 0.293 0.29 1.129 0.456
IGR-39 gCSI 50.484 0.126 0.101 16.095 0.472
IPC-298 gCSI 51.091 0.191 0.181 4.571 0.485
MEL-HO gCSI 50.430 0.238 0.238 0.000 0.484
MEL-JUSO gCSI 54.057 0.171 0.171 0.000 0.5
Mewo gCSI 42.149 0.476 0.462 1.891 0.388
RPMI-7951 gCSI 56.168 0.133 0.129 2.094 0.529
RVH-421 gCSI 43.968 0.42 0.42 0.000 0.418
SK-MEL-1 gCSI 30.456 0.969 0.893 13.936 0.289
SK-MEL-2 gCSI 31.098 1.3 1.3 0.000 0.301
SK-MEL-24 gCSI 42.427 0.371 0.271 13.384 0.379
SK-MEL-3 gCSI 37.714 0.728 0.728 0.000 0.358
SK-MEL-30 gCSI 50.068 0.246 0.246 0.000 0.469
WM-115 gCSI 35.796 0.677 0.603 10.200 0.333
WM-266-4 gCSI 61.738 0.0839 0.0839 0.000 0.578
RPMI-7951 CTRPv2 58.738 0.133 0.13 1.924 0.563
A375 CTRPv2 51.794 0.27 0.265 2.328 0.504
MEL-HO CTRPv2 54.101 0.213 0.208 2.279 0.522
SK-MEL-1 CTRPv2 44.927 0.511 0.473 5.362 0.423
Hs 944.T CTRPv2 66.051 0.0535 0.0497 2.489 0.623
MEL-JUSO CTRPv2 44.173 0.58 0.548 4.093 0.417
SK-MEL-31 CTRPv2 33.742 1.39 1.13 13.704 0.31
SK-MEL-5 CTRPv2 46.095 0.549 0.549 0.000 0.424
IPC-298 CTRPv2 51.206 0.302 0.292 1.666 0.48
SK-MEL-30 CTRPv2 42.407 0.742 0.725 2.213 0.404
A375 CTRPv2 48.798 0.392 0.384 1.367 0.462
WM1799 CTRPv2 46.794 0.297 0.247 12.866 0.44
WM-793 CTRPv2 53.604 0.246 0.246 0.000 0.495
G-361 CTRPv2 55.526 0.202 0.202 0.000 0.517
Hs 852.T CTRPv2 56.318 0.182 0.182 0.000 0.52
Hs 936.T CTRPv2 51.762 0.301 0.301 0.000 0.477
COLO-800 CTRPv2 48.979 0.383 0.362 2.084 0.446
K029AX CTRPv2 41.617 0.588 0.588 0.000 0.379
COLO-829 CTRPv2 52.323 0.272 0.272 0.000 0.47
IGR-1 CTRPv2 47.807 0.459 0.459 0.000 0.439
SH-4 CTRPv2 29.902 1.59 1.39 8.523 0.271
HT-144 CTRPv2 46.172 0.494 0.475 2.642 0.436
Hs 294T CTRPv2 55.525 0.204 0.204 0.000 0.528
SK-MEL-2 CTRPv2 32.322 2.15 2.13 2.058 0.314
A101D CTRPv2 47.300 0.399 0.383 4.413 0.456
A2058 CTRPv2 50.717 0.199 0.188 9.978 0.493
COLO-792 CTRPv2 31.710 2.44 2.44 0.000 0.308
HMCB CTRPv2 41.422 0.894 0.894 0.000 0.382
IGR-39 CTRPv2 46.706 0.265 0.0757 26.668 0.409
Mewo CTRPv2 43.779 0.662 0.629 2.312 0.4
WM-115 CTRPv2 56.782 0.175 0.173 0.542 0.542
WM-266-4 CTRPv2 55.329 0.209 0.209 0.000 0.532
Hs 895.T CTRPv2 30.749 2.16 0.84 27.099 0.258
SK-MEL-24 CTRPv2 35.011 0.644 0.344 30.687 0.313
RVH-421 CTRPv2 40.119 1.02 1.02 0.000 0.379
Hs 839.T CTRPv2 37.607 1.36 1.34 0.831 0.334
WM-88 CTRPv2 52.279 0.285 0.285 0.000 0.483
WM-983B CTRPv2 36.280 1.08 0.889 12.377 0.335
CJM CTRPv2 45.934 0.557 0.557 0.000 0.425
SK-MEL-3 CTRPv2 37.047 1.4 1.4 0.000 0.345
IGR-37 CTRPv2 48.575 0.356 0.342 3.978 0.467
Hs 934.T CTRPv2 28.587 24.6 24.6 0.000 0.207
Hs 688(A).T CTRPv2 19.769 12.3 12.3 0.000 0.153
Hs 940.T CTRPv2 49.728 0.28 0.232 8.351 0.458
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