Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
HDQ-P1 GDSC1000 16.780 0.0122 0.00231 46.233 0.12
HCC2218 GDSC1000 1.917 N/A 0.0242 54.583 0
MDA-MB-231 GDSC1000 24.951 0.0248 0.000848 48.731 0.181
CAL-51 GDSC1000 26.650 0.00329 0.00276 9.511 0.214
MDA-MB-468 GDSC1000 21.967 0.00511 0.003 22.726 0.164
Hs-578-T GDSC1000 27.391 0.00335 0.00314 3.272 0.218
EFM-19 GDSC1000 48.756 0.000945 0.000945 0.000 0.431
HCC70 GDSC1000 43.508 0.00478 0.00478 0.000 0.372
T47D GDSC1000 23.990 0.00223 0.00169 33.459 0.212
CAL-120 GDSC1000 27.534 0.0038 0.003 9.333 0.211
MRK-nu-1 GDSC1000 4.123 85.3 85.3 0.000 0
BT-483 GDSC1000 1.001 N/A 0.0285 97.998 0
EVSA-T GDSC1000 33.691 0.00186 0.0009 29.251 0.277
MCF7 GDSC1000 40.839 0.00173 0.000688 20.742 0.343
MDA-MB-436 GDSC1000 19.841 0.0078 0.00381 24.794 0.137
MFM-223 GDSC1000 27.240 0.00491 0.00491 0.000 0.2
MDA-MB-453 GDSC1000 22.763 0.00254 0.00123 45.600 0.191
BT-20 GDSC1000 35.167 0.00493 0.00493 0.000 0.28
HCC1500 GDSC1000 7.421 N/A 0.000104 85.158 0
OCUB-M GDSC1000 26.056 0.00459 0.00176 30.257 0.195
HCC2157 GDSC1000 24.185 0.00366 0.00273 16.357 0.194
DU-4475 GDSC1000 8.586 0.0249 0.01 32.812 0.0428
COLO-824 GDSC1000 20.227 0.00763 0.00763 0.000 0.137
HCC1937 GDSC1000 19.984 0.0307 0.0307 0.000 0
JIMT-1 GDSC1000 47.174 0.000849 0.000643 10.924 0.413
BT-474 GDSC1000 6.706 0.0141 0.0141 0.000 0
MDA-MB-175-VII GDSC1000 6.613 N/A 0.00964 54.716 0.022
CAL-85-1 GDSC1000 23.093 0.00547 0.00547 0.000 0.167
HCC1419 GDSC1000 3.933 N/A 0.00623 76.773 0.00626
AU565 GDSC1000 33.601 0.00202 0.00161 11.710 0.281
EFM-192A GDSC1000 12.794 0.0269 0.00991 27.336 0.0667
HCC1569 GDSC1000 7.723 N/A 0.000278 88.146 0.00315
ZR-75-30 GDSC1000 10.662 0.0127 0.0127 0.000 0
HCC1187 GDSC1000 42.480 0.00117 0.000658 19.136 0.361
MDA-MB-361 GDSC1000 22.451 0.00325 0.00303 12.113 0.205
HARA GDSC1000 50.981 0.000675 0.000555 7.132 0.455
BT-549 GDSC1000 35.936 0.0033 0.000907 25.547 0.288
HCC1395 GDSC1000 9.484 0.0149 0.00628 38.266 0.0589
HCC1954 GDSC1000 17.264 N/A 0.00122 59.829 0.103
HCC38 GDSC1000 16.689 0.00759 0.00759 0.000 0.115
UACC-893 GDSC1000 7.806 N/A 0.00282 70.916 0.0475
HCC1143 GDSC1000 26.238 0.00238 0.00138 34.123 0.221
HCC1428 GDSC1000 10.869 0.0926 0.0272 25.411 0
MDA-MB-330 GDSC1000 10.174 N/A 0.0054 60.273 0.0361
HCC202 GDSC1000 1.475 N/A 0.00409 92.695 0
MDA-MB-415 GDSC1000 30.972 0.00302 0.00184 17.257 0.243
AU565 gCSI 32.255 0.01 0.00888 19.529 0.304
BT-20 gCSI 35.797 0.00822 0.00612 19.239 0.325
BT-474 gCSI 19.569 0.0347 0.0218 34.414 0.17
BT-549 gCSI 43.771 0.00433 0.00339 14.245 0.401
CAL-120 gCSI 23.059 0.0263 0.0122 36.837 0.196
CAL-148 gCSI 36.136 0.00747 0.00656 16.966 0.341
CAL-51 gCSI 39.607 0.00734 0.00634 9.838 0.365
CAMA-1 gCSI 16.773 N/A 0.0148 51.019 0.14
EFM-19 gCSI 31.332 0.0147 0.013 12.403 0.291
EVSA-T gCSI 35.814 0.00438 0.00343 29.652 0.331
HCC1143 gCSI 33.732 0.00755 0.00454 29.322 0.301
HCC1187 gCSI 42.684 0.00676 0.00655 2.063 0.395
HCC1419 gCSI 0.439 N/A 0.000178 99.122 0
HCC1806 gCSI 40.334 0.00613 0.00561 10.984 0.383
HCC1937 gCSI 8.617 N/A 0.00969 77.963 0.0408
HCC1954 gCSI 42.614 0.00533 0.0041 12.845 0.385
HCC38 gCSI 32.028 0.00893 0.00272 40.180 0.272
HDQ-P1 gCSI 19.627 0.0313 0.00988 49.502 0.167
Hs-578-T gCSI 45.518 0.00401 0.00335 11.032 0.421
MCF7 gCSI 21.656 0.0319 0.0104 43.429 0.18
MDA-MB-157 gCSI 30.044 0.0169 0.0154 11.153 0.282
MDA-MB-175-VII gCSI 2.903 N/A 0.0291 89.080 0.00172
MDA-MB-231 gCSI 25.443 0.0238 0.00737 39.770 0.211
MDA-MB-436 gCSI 31.717 0.0112 0.00548 30.456 0.274
MDA-MB-453 gCSI 11.986 N/A 0.00743 71.537 0.0789
MDA-MB-468 gCSI 41.100 0.00424 0.00352 18.799 0.385
MFM-223 gCSI 41.051 0.00435 0.00316 20.814 0.376
SK-BR-3 gCSI 20.262 0.0391 0.0165 38.726 0.168
T47D gCSI 20.473 N/A 0.00685 52.434 0.162
184A1 GRAY 18.011 N/A 0.00556 69.042 0.119
184B5 GRAY 16.976 N/A 1.09e-05 76.505 0.0775
AU565 GRAY 52.906 0.00182 0.0015 22.634 0.504
BT-549 GRAY 52.373 0.0027 0.00162 22.660 0.485
HCC1187 GRAY 52.607 0.00921 0.00846 4.239 0.497
HCC1569 GRAY 27.705 N/A 0.00353 55.131 0.229
HCC1806 GRAY 62.357 0.00153 0.00139 9.565 0.605
HCC2185 GRAY 13.911 N/A 0.00239 78.242 0.0624
HCC3153 GRAY 32.004 0.0329 0.00969 40.617 0.279
HCC70 GRAY 35.088 0.0175 0.00642 38.537 0.31
MCF10A GRAY 53.556 0.00391 0.00249 16.744 0.496
MCF12A GRAY 44.171 0.00722 0.00159 34.605 0.387
MDA-MB-231 GRAY 63.909 0.00134 0.00115 9.193 0.612
MDA-MB-361 GRAY 23.294 N/A 0.0105 56.267 0.189
MDA-MB-415 GRAY 14.262 N/A 0.0155 71.616 0.0946
MDA-MB-453 GRAY 31.026 0.0383 0.0104 41.806 0.269
SK-BR-3 GRAY 37.316 0.0174 0.0143 26.610 0.352
SUM 159PT GRAY 67.013 0.000668 0.000599 11.262 0.649
SUM 159PT GRAY 64.612 0.00106 0.000917 10.508 0.622
SUM 229PE GRAY 34.419 0.0214 0.0102 35.659 0.309
SUM 229PE GRAY 32.516 0.036 0.013 36.967 0.286
SUM 52PE GRAY 28.979 N/A 0.00181 53.912 0.211
T47D GRAY 29.624 N/A 0.00363 51.853 0.251
T47D_KBluc GRAY 27.883 0.0533 0.0168 43.788 0.242
UACC-812 GRAY 23.744 N/A 0.0077 57.355 0.196
184A1 GRAY 12.578 N/A 0.0111 76.203 0.0715
184A1 GRAY 13.609 N/A 0.00293 78.430 0.0678
184A1 GRAY 8.968 N/A 0.00229 86.215 0.021
184B5 GRAY 21.091 N/A 0.00184 68.411 0.145
600MPE GRAY 6.807 N/A 0.0309 84.979 0.00975
600MPE GRAY 8.111 N/A 0.0374 81.316 0.0371
600MPE GRAY 12.304 N/A 0.0239 73.756 0.0776
AU565 GRAY 51.251 0.00604 0.00556 11.965 0.497
AU565 GRAY 52.728 0.00742 0.00706 6.440 0.513
BT-474 GRAY 35.285 0.0115 0.00769 36.637 0.323
BT-474 GRAY 28.508 0.0416 0.00818 48.365 0.245
BT-474 GRAY 29.040 0.0233 0.0143 42.900 0.26
BT-483 GRAY 14.076 N/A 0.0204 70.745 0.0989
BT-483 GRAY 10.659 N/A 0.033 75.987 0.0588
BT-549 GRAY 41.574 0.00604 0.00343 32.907 0.38
CAMA-1 GRAY 33.864 0.0086 0.00544 41.991 0.306
HBL-100 GRAY 47.261 0.00215 0.00155 30.623 0.441
HBL-100 GRAY 47.241 0.00157 0.000977 34.126 0.435
HBL-100 GRAY 45.930 0.0021 0.00122 34.400 0.421
HCC1143 GRAY 40.880 0.0156 0.00574 29.395 0.362
HCC1143 GRAY 27.881 0.0588 0.0208 41.877 0.243
HCC1187 GRAY 54.097 0.00476 0.00392 11.193 0.513
HCC1187 GRAY 48.871 0.0116 0.0102 8.632 0.465
HCC1187 GRAY 52.333 0.00938 0.00843 4.770 0.491
HCC1395 GRAY 35.254 0.0175 0.0107 33.603 0.322
HCC1395 GRAY 29.647 0.0145 0.00659 47.886 0.261
HCC1395 GRAY 22.618 N/A 0.00959 58.099 0.186
HCC1419 GRAY 9.741 N/A 0.0176 80.223 0.0506
HCC1419 GRAY 6.223 N/A 0.0678 83.956 0.0238
HCC1419 GRAY 13.699 N/A 0.0168 72.399 0.088
HCC1419 GRAY 6.607 N/A 0.0555 83.622 0.0257
HCC1428 GRAY 6.572 N/A 0.0155 86.917 0.0115
HCC1428 GRAY 6.506 N/A 0.0171 86.855 0.0134
HCC1428 GRAY 15.218 N/A 0.005 74.205 0.0885
HCC1569 GRAY 21.456 N/A 0.00288 66.110 0.164
HCC1806 GRAY 58.739 0.0026 0.00246 8.977 0.574
HCC1806 GRAY 41.787 0.00614 0.00279 34.261 0.377
HCC1806 GRAY 57.361 0.00284 0.00258 10.604 0.555
HCC1937 GRAY 19.712 N/A 0.00475 66.837 0.149
HCC1954 GRAY 62.453 0.00223 0.00204 5.328 0.599
HCC1954 GRAY 57.348 0.00367 0.00323 8.123 0.548
HCC1954 GRAY 57.324 0.00299 0.00236 11.553 0.541
HCC202 GRAY 22.971 N/A 0.0106 56.810 0.185
HCC202 GRAY 27.921 0.338 0.0103 47.748 0.226
HCC2185 GRAY 23.096 N/A 0.002 65.075 0.169
HCC2185 GRAY 23.581 N/A 0.00398 61.217 0.19
HCC2185 GRAY 19.402 N/A 0.00453 67.544 0.134
HCC2185 GRAY 18.520 N/A 0.00364 69.889 0.128
HCC2185 GRAY 8.388 N/A 0.00114 88.105 0.0137
HCC3153 GRAY 18.032 N/A 0.0105 66.157 0.127
HCC3153 GRAY 32.532 0.0326 0.016 34.966 0.292
HCC38 GRAY 31.945 N/A 0.00028 60.766 0.26
HCC38 GRAY 45.013 0.00601 0.00356 26.996 0.415
HCC38 GRAY 51.245 0.00262 0.00211 22.032 0.487
HCC70 GRAY 38.855 0.0133 0.00778 30.112 0.356
HCC70 GRAY 45.496 0.00863 0.00492 23.072 0.417
Hs-578-T GRAY 52.888 0.00378 0.00259 17.490 0.494
Hs-578-T GRAY 50.672 0.00266 0.00193 23.703 0.477
LY2 GRAY 43.158 0.00782 0.00459 27.703 0.397
LY2 GRAY 27.261 N/A 0.00759 51.140 0.228
MCF10A GRAY 50.453 0.00341 0.00208 23.352 0.467
MCF10A GRAY 56.846 0.00273 0.00225 12.842 0.542
MCF10A GRAY 51.005 0.00301 0.00198 22.970 0.476
MCF10F GRAY 44.753 0.00377 0.00217 31.688 0.411
MCF12A GRAY 47.404 0.00273 0.00193 28.616 0.443
MCF12A GRAY 26.468 N/A 0.00519 54.928 0.21
MCF7 GRAY 28.387 0.144 0.00892 47.949 0.236
MCF7 GRAY 15.942 N/A 0.0155 68.261 0.111
MCF7 GRAY 36.629 0.0209 0.00566 36.891 0.319
MDA-MB-134-VI GRAY 35.135 0.0149 0.00712 37.576 0.315
MDA-MB-134-VI GRAY 12.955 N/A 0.0154 74.218 0.054
MDA-MB-134-VI GRAY 7.862 N/A 0.0242 83.198 0.0329
MDA-MB-157 GRAY 47.136 0.00889 0.00681 16.778 0.444
MDA-MB-157 GRAY 51.984 0.00442 0.00338 16.257 0.491
MDA-MB-175-VII GRAY 12.709 N/A 0.00948 76.494 0.0777
MDA-MB-175-VII GRAY 13.356 N/A 0.00495 77.409 0.077
MDA-MB-231 GRAY 48.363 0.00277 0.00231 25.617 0.459
MDA-MB-231 GRAY 51.977 0.00366 0.00272 18.470 0.49
MDA-MB-231 GRAY 55.972 0.00164 0.00126 19.729 0.531
MDA-MB-361 GRAY 29.221 0.0235 0.0138 42.883 0.262
MDA-MB-361 GRAY 25.542 N/A 0.00691 54.806 0.209
MDA-MB-361 GRAY 31.608 0.0428 0.00398 48.019 0.268
MDA-MB-415 GRAY 27.292 N/A 0.00226 58.130 0.215
MDA-MB-415 GRAY 28.211 N/A 0.00371 54.018 0.23
MDA-MB-436 GRAY 25.191 0.0438 0.0191 48.191 0.22
MDA-MB-436 GRAY 25.898 N/A 0.00696 54.106 0.203
MDA-MB-436 GRAY 13.545 8.43 0.868 37.313 0.0902
MDA-MB-436 GRAY 22.279 N/A 0.00992 58.521 0.177
MDA-MB-453 GRAY 7.778 N/A 0.0151 84.536 0.00466
MDA-MB-453 GRAY 45.905 0.00558 0.00418 24.026 0.432
MDA-MB-453 GRAY 36.444 0.0259 0.0048 38.517 0.313
MDA-MB-453 GRAY 31.676 0.0295 0.0135 38.272 0.282
MDA-MB-468 GRAY 58.260 0.00305 0.00259 9.147 0.554
MDA-MB-468 GRAY 52.897 0.00275 0.00149 22.561 0.487
MDA-MB-468 GRAY 55.198 0.00504 0.00419 8.562 0.52
MDA-MB-468 GRAY 47.385 0.0106 0.00995 11.745 0.46
S1 GRAY 41.054 0.00964 0.00436 31.687 0.37
SK-BR-3 GRAY 44.894 0.0102 0.00763 19.472 0.422
SK-BR-3 GRAY 32.651 0.029 0.0196 32.563 0.3
SK-BR-3 GRAY 45.533 0.013 0.0104 14.664 0.429
SUM102PT GRAY 13.468 8.66e+03 8.66e+03 0.000 0
SUM 1315M02 GRAY 32.867 0.0862 0.0203 31.796 0.277
SUM 1315M02 GRAY 37.646 0.0178 0.00804 31.969 0.338
SUM 1315M02 GRAY 47.730 0.00998 0.00528 18.303 0.431
SUM 149PT GRAY 51.329 0.00172 0.0011 27.468 0.478
SUM 159PT GRAY 55.449 0.00303 0.00282 12.661 0.539
SUM 159PT GRAY 47.053 0.0115 0.0108 11.347 0.457
SUM185PE GRAY 18.997 N/A 0.0173 61.550 0.151
SUM185PE GRAY 13.946 N/A 0.0152 72.318 0.0951
SUM 229PE GRAY 43.379 0.00575 0.00373 29.240 0.402
SUM 52PE GRAY 47.862 0.00271 0.00189 28.146 0.447
SUM 52PE GRAY 46.292 0.00494 0.00272 27.374 0.425
T47D GRAY 28.170 N/A 0.00309 55.121 0.238
T4 GRAY 55.532 0.00253 0.00199 16.095 0.527
UACC-812 GRAY 18.975 N/A 0.00333 69.490 0.135
UACC-812 GRAY 18.422 N/A 0.00309 70.655 0.131
UACC-812 GRAY 16.561 N/A 0.00284 73.887 0.11
UACC-812 GRAY 18.066 N/A 0.00915 66.754 0.136
UACC-893 GRAY 28.613 0.0295 0.0192 41.121 0.258
UACC-893 GRAY 4.412 6.63e+03 6.63e+03 0.000 0
UACC-893 GRAY 5.657 7.99e+04 7.99e+04 0.000 0
UACC-893 GRAY 17.745 N/A 0.0223 62.584 0.136
UACC-893 GRAY 25.768 0.0382 0.016 48.460 0.225
UACC-893 GRAY 13.306 N/A 0.04 68.974 0.0919
ZR-75-1 GRAY 42.296 0.0174 0.0121 18.974 0.392
ZR-75-1 GRAY 14.219 N/A 0.00397 76.615 0.0792
ZR-75-1 GRAY 11.015 N/A 0.00624 80.781 0.0513
ZR-75-30 GRAY 10.128 N/A 0.00465 83.007 0.0438
ZR75B GRAY 13.901 N/A 0.0132 73.005 0.089
ZR75B GRAY 24.502 N/A 0.00264 61.718 0.192
HCC1428 CTRPv2 12.575 2.52e+03 2.52e+03 0.000 0
HCC38 CTRPv2 59.923 0.00742 0.000466 32.473 0.555
BT-549 CTRPv2 66.147 0.0014 0.00067 32.991 0.624
HCC202 CTRPv2 41.063 16.9 16.9 0.000 0.345
DU-4475 CTRPv2 83.659 0.00283 0.00245 3.849 0.818
HCC1500 CTRPv2 39.613 3.67 3.67 0.000 0.329
Hs-578-T CTRPv2 69.983 0.000315 5.49e-05 12.654 0.666
MDA-MB-468 CTRPv2 73.294 1.05e-05 1e-06 23.780 0.703
CAL-85-1 CTRPv2 72.539 0.000844 0.000325 25.156 0.695
BT-20 CTRPv2 64.032 0.00184 0.000338 33.221 0.6
HCC1419 CTRPv2 24.386 29.2 29.2 0.000 0.167
ZR-75-30 CTRPv2 25.042 1.09e+11 1e+06 22.178 0
EFM-192A CTRPv2 65.107 0.0112 0.00388 24.083 0.612
MDA-MB-157 CTRPv2 71.477 0.00245 0.000888 22.337 0.683
MDA-MB-361 CTRPv2 25.899 N/A 1e-06 74.101 0.177
T47D CTRPv2 23.679 N/A 0.00381 74.535 0.153
BT-474 CTRPv2 45.132 0.0256 0.011 46.001 0.399
HCC2218 CTRPv2 19.429 N/A 0.323 62.008 0.153
SK-BR-3 CTRPv2 69.259 0.00585 0.00491 24.130 0.66
MDA-MB-453 CTRPv2 47.519 0.0272 0.0034 49.121 0.417
AU565 CTRPv2 69.592 0.00354 0.00215 27.038 0.662
MDA-MB-415 CTRPv2 24.305 8.11e+08 2.66e+04 24.849 0
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