Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A101D GDSC1000 32.483 N/A 0.0194 56.992 0.265
GAK GDSC1000 0.632 2.06 2.06 0.000 0
MKL-1-subclone-2 GDSC1000 4.273 N/A 0.161 91.454 0
DJM-1 GDSC1000 3.925 3.16 3.16 0.000 0
MZ7-mel GDSC1000 28.757 0.166 0.132 29.807 0.26
IST-MEL1 GDSC1000 46.231 0.0935 0.0248 28.384 0.403
MZ2-MEL GDSC1000 34.255 0.247 0.247 0.000 0.276
A253 GDSC1000 19.128 10.6 10.6 0.000 0
HT-144 GDSC1000 37.528 0.985 0.0164 48.946 0.306
CP66-MEL GDSC1000 31.517 0.168 0.132 22.988 0.282
SK-MEL-2 GDSC1000 14.864 N/A 0.00456 84.776 0.0541
CP67-MEL GDSC1000 37.968 0.207 0.179 4.573 0.311
COLO-800 GDSC1000 9.063 N/A 0.0222 86.000 0.00754
LB2518-MEL GDSC1000 39.659 0.142 0.133 4.098 0.347
MMAC-SF GDSC1000 3.261 2.97 2.97 0.000 0
COLO-829 GDSC1000 50.934 0.0524 0.0484 13.782 0.485
LB373-MEL-D GDSC1000 16.181 0.8 0.8 0.000 0.111
SH-4 GDSC1000 36.297 0.202 0.202 0.000 0.3
SK-MEL-1 GDSC1000 2.500 N/A 31.6 95.000 0
A388 GDSC1000 54.418 0.0494 0.0381 12.179 0.494
MKL-2 GDSC1000 2.746 N/A 0.187 94.509 0
RPMI-7951 CTRPv2 40.495 1.24 1.24 0.000 0.342
A375 CTRPv2 20.547 7.04 6.67 6.733 0.191
MEL-HO CTRPv2 16.675 12.2 12.2 0.000 0.144
SK-MEL-1 CTRPv2 12.348 18.9 18.9 0.000 0.107
Hs 944.T CTRPv2 13.055 18.1 18.1 0.000 0.11
MEL-JUSO CTRPv2 13.291 16.6 16.6 0.000 0.121
SK-MEL-31 CTRPv2 9.247 31.7 31.7 0.000 0.0695
SK-MEL-5 CTRPv2 10.560 22.1 22.1 0.000 0.097
IPC-298 CTRPv2 10.613 21.6 21 4.242 0.0949
SK-MEL-30 CTRPv2 6.864 32.8 32.8 0.000 0.0601
A375 CTRPv2 23.072 13.8 13.8 0.000 0.168
WM1799 CTRPv2 13.008 17.9 17.9 0.000 0.112
WM-793 CTRPv2 33.679 3.28 3.28 0.000 0.27
G-361 CTRPv2 11.492 11.2 11 2.365 0.0977
Hs 852.T CTRPv2 47.509 0.211 0.014 36.888 0.417
Hs 936.T CTRPv2 4.748 26.5 19.1 27.888 0.0331
COLO-800 CTRPv2 9.843 28.5 28.5 0.000 0.0761
K029AX CTRPv2 13.113 22.4 22.4 0.000 0.0999
COLO-829 CTRPv2 38.527 14.7 14.7 0.000 0.317
IGR-1 CTRPv2 13.262 19.1 19.1 0.000 0.107
SH-4 CTRPv2 23.924 8.46 8.46 0.000 0.186
A253 CTRPv2 5.455 80.8 80.8 0.000 0
C32 CTRPv2 6.432 42.7 42.7 0.000 0.0462
HT-144 CTRPv2 13.825 16.7 16.7 0.000 0.117
Hs 294T CTRPv2 21.209 8.28 8.28 0.000 0.178
A101D CTRPv2 28.515 10.4 10.4 0.000 0.211
A2058 CTRPv2 5.734 37.2 37.2 0.000 0.0489
COLO-792 CTRPv2 7.246 31.6 31.6 0.000 0.0634
HMCB CTRPv2 13.503 18.8 18.8 0.000 0.109
IGR-39 CTRPv2 64.269 0.0097 0.00317 26.982 0.603
Mewo CTRPv2 26.371 9.74 9.74 0.000 0.196
WM-115 CTRPv2 37.486 1.56 1.56 0.000 0.32
WM-266-4 CTRPv2 15.664 14.8 14.8 0.000 0.128
Hs 895.T CTRPv2 42.694 2.2 2.2 0.000 0.363
SK-MEL-24 CTRPv2 39.130 1.78 1.78 0.000 0.324
RVH-421 CTRPv2 14.748 17.4 17.4 0.000 0.117
Hs 839.T CTRPv2 49.674 0.191 0.0101 32.539 0.441
WM-88 CTRPv2 18.420 8.64 7.29 13.370 0.163
WM-983B CTRPv2 44.214 0.724 0.154 20.935 0.38
CJM CTRPv2 27.893 5.38 5.38 0.000 0.222
SK-MEL-3 CTRPv2 18.475 19.7 19.7 0.000 0.132
IGR-37 CTRPv2 14.648 20.9 20.9 0.000 0.11
Hs 934.T CTRPv2 47.968 0.0578 0.00494 45.410 0.422
Hs 688(A).T CTRPv2 25.488 54.3 54.3 0.000 0.173
Hs 940.T CTRPv2 39.513 1.97 1.97 0.000 0.328
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