Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A2058 CCLE 2.479 8.2 8.2 0.000 0
A253 CCLE 1.678 12.3 12.1 2.091 0
A375 CCLE 5.335 5.81 5.81 0.000 0.0397
C32 CCLE 1.382 9.24 9.24 0.000 0
CHL-1 CCLE 0.964 11.1 10 16.562 0
COLO-679 CCLE 1.581 8.85 8.85 0.000 0
G-361 CCLE 4.606 5.88 5.88 0.000 0.0358
HMCB CCLE 3.203 8 8 0.000 0
Hs 294T CCLE 7.506 N/A 2.29 51.664 0.0577
Hs 695T CCLE 1.382 9.24 9.24 0.000 0
Hs 852.T CCLE 8.323 4.88 4.88 0.000 0.0619
Hs 895.T CCLE 6.024 5.86 5.86 0.000 0.043
Hs 936.T CCLE 0.809 10.8 10.8 0.000 0
Hs 939.T CCLE 1.461 N/A 2.79 88.837 0.000459
Hs 944.T CCLE 5.954 5.84 3.41 44.222 0.0454
HT-144 CCLE 2.147 8.37 8.37 0.000 0
IGR-37 CCLE 5.260 N/A 3.06 56.080 0.0371
IGR-39 CCLE 6.959 7.35 7.35 0.000 0.0427
IPC-298 CCLE 0.691 11.3 11.3 0.000 0
K029AX CCLE 2.539 7.54 7.54 0.000 0.0162
MEL-HO CCLE 5.281 5.49 5.49 0.000 0.0423
Mewo CCLE 1.061 10 10 0.000 0
RPMI-7951 CCLE 6.684 5.07 3.14 42.670 0.0523
RVH-421 CCLE 0.467 12.6 12.6 0.000 0
SF8657 CCLE 1.268 10 10 0.000 0
SK-MEL-2 CCLE 1.812 N/A 3.72 96.375 0
SK-MEL-24 CCLE 1.530 8.95 8.95 0.000 0
SK-MEL-30 CCLE 0.809 10.8 10.8 0.000 0
SK-MEL-31 CCLE 2.609 7.46 7.46 0.000 0.0168
SK-MEL-5 CCLE 1.530 8.95 8.95 0.000 0
WM-115 CCLE 2.254 N/A 0.405 93.901 0
WM1799 CCLE 1.240 9.55 9.55 0.000 0
WM-266-4 CCLE 5.546 N/A 2.58 60.577 0.0383
WM-793 CCLE 3.142 8.25 8.25 0.000 0
WM-88 CCLE 3.192 8.56 8.56 0.000 0
WM-983B CCLE 6.581 5.85 5.85 0.000 0.0462
A101D GDSC1000 6.003 1.41e+04 1.41e+04 0.000 0
MMAC-SF GDSC1000 0.636 3.21 3.21 0.000 0
IST-MEL1 GDSC1000 7.508 N/A 0.00395 84.984 0
MKL-1-subclone-2 GDSC1000 7.996 N/A 0.0645 84.007 0
MZ7-mel GDSC1000 4.492 N/A 2.63 91.016 0
COLO-800 GDSC1000 5.261 N/A 1.25e+03 89.478 0
COLO-829 GDSC1000 4.657 N/A 1e+06 90.687 0
MKL-2 GDSC1000 7.693 258 258 0.000 0
CP67-MEL GDSC1000 15.083 N/A 1e+06 69.833 0
LB373-MEL-D GDSC1000 0.355 3.74 3.74 0.000 0
LB2518-MEL GDSC1000 9.665 N/A 0.000186 80.670 0
CP66-MEL GDSC1000 3.745 N/A 324 92.510 0
GAK GDSC1000 8.084 N/A 1e+06 83.832 0
SK-MEL-2 GDSC1000 3.998 N/A 0.153 91.667 0
MZ2-MEL GDSC1000 6.230 N/A 161 87.539 0
A253 GDSC1000 4.265 N/A 8.5e+05 90.259 0
HT-144 GDSC1000 8.847 N/A 15.2 82.306 0
DJM-1 GDSC1000 5.242 N/A 0.013 89.515 0
SH-4 GDSC1000 10.224 N/A 13.7 79.553 0
SK-MEL-1 GDSC1000 4.063 N/A 0.011 95.623 0
A388 GDSC1000 6.611 73 73 0.000 0
A2058 gCSI 2.383 2.05 2.05 0.000 0
A375 gCSI 3.407 0.901 0.901 0.000 0.0221
A388 gCSI 28.217 1.69 1.69 0.000 0.259
A431 gCSI 0.432 1.57 1.57 0.000 0
C32 gCSI 4.737 1.3e+03 1.3e+03 0.000 0
CHL-1 gCSI 6.893 N/A 0.00349 89.082 0.00141
COLO-679 gCSI 4.650 N/A 0.0078 91.226 0
COLO-800 gCSI 7.074 N/A 0.0358 83.200 0.00432
COLO-829 gCSI 6.760 1.42 1.42 0.000 0
G-361 gCSI 8.489 7.51 7.51 0.000 0
HMV-II gCSI 9.858 8.43e+06 1e+06 10.974 0
Hs 294T gCSI 2.584 1.15 1.15 0.000 0
Hs 695T gCSI 3.128 N/A 0.491 71.341 0.0081
Hs 852.T gCSI 4.172 3.44 3.44 0.000 0
IGR-1 gCSI 3.658 0.965 0.965 0.000 0.0222
IGR-37 gCSI 4.845 6.97 6.97 0.000 0
IGR-39 gCSI 3.907 N/A 0.263 74.351 0.0201
IPC-298 gCSI 2.081 5.73 5.73 0.000 0
MEL-HO gCSI 10.364 567 567 0.000 0
MEL-JUSO gCSI 1.016 1.24 1.24 0.000 0
Mewo gCSI 9.914 153 153 0.000 0
RPMI-7951 gCSI 2.303 3.8 3.8 0.000 0
RVH-421 gCSI 3.218 5.79 5.79 0.000 0
SK-MEL-1 gCSI 2.569 1.44e+05 1.44e+05 0.000 0
SK-MEL-2 gCSI 5.816 N/A 0.00393 88.369 0
SK-MEL-24 gCSI 4.262 6.05 6.05 0.000 0
SK-MEL-3 gCSI 3.105 4.7 4.7 0.000 0
SK-MEL-30 gCSI 6.691 40.5 40.5 0.000 0
WM-115 gCSI 6.362 9.98e+04 9.98e+04 0.000 0
WM-266-4 gCSI 4.750 N/A 0.335 61.930 0.032
A375 CTRPv2 25.195 4.75 4.73 0.581 0.239
MEL-HO CTRPv2 25.007 4.88 4.88 0.113 0.241
SK-MEL-1 CTRPv2 21.469 6.78 6.69 2.444 0.205
Hs 944.T CTRPv2 23.800 5.79 5.79 0.000 0.21
MEL-JUSO CTRPv2 22.859 6.14 6.14 0.000 0.212
SK-MEL-31 CTRPv2 16.873 11.5 11.5 0.000 0.153
SK-MEL-5 CTRPv2 17.059 11.2 11.2 0.000 0.162
IPC-298 CTRPv2 19.723 8.49 8.49 0.000 0.185
SK-MEL-30 CTRPv2 17.674 10.5 10.5 0.000 0.168
A375 CTRPv2 17.264 11.1 11.1 0.000 0.155
WM1799 CTRPv2 20.680 7.86 7.86 0.000 0.185
WM-793 CTRPv2 18.553 9.79 9.79 0.000 0.165
G-361 CTRPv2 20.310 7.82 7.58 2.810 0.184
Hs 852.T CTRPv2 28.666 2.09 1.87 16.261 0.271
Hs 936.T CTRPv2 18.215 14.3 14.3 0.000 0.14
COLO-800 CTRPv2 17.671 5.45 5.26 6.556 0.166
K029AX CTRPv2 19.174 5.13 5.13 0.000 0.182
COLO-829 CTRPv2 26.323 4.45 4.45 0.000 0.233
IGR-1 CTRPv2 28.356 3.02 2.94 5.162 0.273
SH-4 CTRPv2 29.498 2.99 2.97 1.027 0.286
A253 CTRPv2 8.476 29.3 29.3 0.000 0.0697
C32 CTRPv2 19.509 8.99 8.99 0.000 0.172
HT-144 CTRPv2 24.598 4.85 4.78 2.503 0.235
Hs 294T CTRPv2 26.477 3.98 3.9 2.637 0.251
SK-MEL-2 CTRPv2 12.747 17.5 17.5 0.000 0.119
A101D CTRPv2 25.276 4.5 4.45 2.513 0.243
A2058 CTRPv2 22.971 5.79 5.73 2.210 0.221
COLO-792 CTRPv2 29.255 2.96 2.92 2.431 0.281
HMCB CTRPv2 9.956 23.5 23.5 0.000 0.0909
IGR-39 CTRPv2 14.034 N/A 3.38 50.855 0.118
Mewo CTRPv2 22.115 6.64 6.38 2.653 0.196
WM-115 CTRPv2 23.743 5.58 5.58 0.000 0.229
WM-266-4 CTRPv2 23.183 5.66 5.6 2.227 0.223
Hs 895.T CTRPv2 22.208 6.67 6.67 0.000 0.2
RVH-421 CTRPv2 22.560 5.98 5.89 2.863 0.216
Hs 839.T CTRPv2 12.214 18.7 18.7 0.000 0.111
WM-88 CTRPv2 21.686 3.28 2.6 30.231 0.199
WM-983B CTRPv2 22.002 5.79 4.68 13.878 0.195
CJM CTRPv2 22.692 5.8 5.7 3.637 0.217
SK-MEL-3 CTRPv2 23.787 5.5 5.48 0.532 0.229
IGR-37 CTRPv2 18.572 9.56 9.56 0.000 0.177
Hs 934.T CTRPv2 25.060 5.09 5.09 0.000 0.221
Hs 688(A).T CTRPv2 25.668 4.69 4.69 0.000 0.23
Hs 940.T CTRPv2 26.427 4.16 4.15 0.630 0.255
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