Summary Statistics
Cell Line | Dataset | AAC (%) | IC50 (µM) | EC50 (µM) | Einf (%) | DSS1 (arb.) |
---|
A2058 | CCLE |
2.479
|
8.2
|
8.2
|
0.000
|
0
|
A253 | CCLE |
1.678
|
12.3
|
12.1
|
2.091
|
0
|
A375 | CCLE |
5.335
|
5.81
|
5.81
|
0.000
|
0.0397
|
C32 | CCLE |
1.382
|
9.24
|
9.24
|
0.000
|
0
|
CHL-1 | CCLE |
0.964
|
11.1
|
10
|
16.562
|
0
|
COLO-679 | CCLE |
1.581
|
8.85
|
8.85
|
0.000
|
0
|
G-361 | CCLE |
4.606
|
5.88
|
5.88
|
0.000
|
0.0358
|
HMCB | CCLE |
3.203
|
8
|
8
|
0.000
|
0
|
Hs 294T | CCLE |
7.506
|
N/A
|
2.29
|
51.664
|
0.0577
|
Hs 695T | CCLE |
1.382
|
9.24
|
9.24
|
0.000
|
0
|
Hs 852.T | CCLE |
8.323
|
4.88
|
4.88
|
0.000
|
0.0619
|
Hs 895.T | CCLE |
6.024
|
5.86
|
5.86
|
0.000
|
0.043
|
Hs 936.T | CCLE |
0.809
|
10.8
|
10.8
|
0.000
|
0
|
Hs 939.T | CCLE |
1.461
|
N/A
|
2.79
|
88.837
|
0.000459
|
Hs 944.T | CCLE |
5.954
|
5.84
|
3.41
|
44.222
|
0.0454
|
HT-144 | CCLE |
2.147
|
8.37
|
8.37
|
0.000
|
0
|
IGR-37 | CCLE |
5.260
|
N/A
|
3.06
|
56.080
|
0.0371
|
IGR-39 | CCLE |
6.959
|
7.35
|
7.35
|
0.000
|
0.0427
|
IPC-298 | CCLE |
0.691
|
11.3
|
11.3
|
0.000
|
0
|
K029AX | CCLE |
2.539
|
7.54
|
7.54
|
0.000
|
0.0162
|
MEL-HO | CCLE |
5.281
|
5.49
|
5.49
|
0.000
|
0.0423
|
Mewo | CCLE |
1.061
|
10
|
10
|
0.000
|
0
|
RPMI-7951 | CCLE |
6.684
|
5.07
|
3.14
|
42.670
|
0.0523
|
RVH-421 | CCLE |
0.467
|
12.6
|
12.6
|
0.000
|
0
|
SF8657 | CCLE |
1.268
|
10
|
10
|
0.000
|
0
|
SK-MEL-2 | CCLE |
1.812
|
N/A
|
3.72
|
96.375
|
0
|
SK-MEL-24 | CCLE |
1.530
|
8.95
|
8.95
|
0.000
|
0
|
SK-MEL-30 | CCLE |
0.809
|
10.8
|
10.8
|
0.000
|
0
|
SK-MEL-31 | CCLE |
2.609
|
7.46
|
7.46
|
0.000
|
0.0168
|
SK-MEL-5 | CCLE |
1.530
|
8.95
|
8.95
|
0.000
|
0
|
WM-115 | CCLE |
2.254
|
N/A
|
0.405
|
93.901
|
0
|
WM1799 | CCLE |
1.240
|
9.55
|
9.55
|
0.000
|
0
|
WM-266-4 | CCLE |
5.546
|
N/A
|
2.58
|
60.577
|
0.0383
|
WM-793 | CCLE |
3.142
|
8.25
|
8.25
|
0.000
|
0
|
WM-88 | CCLE |
3.192
|
8.56
|
8.56
|
0.000
|
0
|
WM-983B | CCLE |
6.581
|
5.85
|
5.85
|
0.000
|
0.0462
|
A101D | GDSC1000 |
6.003
|
1.41e+04
|
1.41e+04
|
0.000
|
0
|
MMAC-SF | GDSC1000 |
0.636
|
3.21
|
3.21
|
0.000
|
0
|
IST-MEL1 | GDSC1000 |
7.508
|
N/A
|
0.00395
|
84.984
|
0
|
MKL-1-subclone-2 | GDSC1000 |
7.996
|
N/A
|
0.0645
|
84.007
|
0
|
MZ7-mel | GDSC1000 |
4.492
|
N/A
|
2.63
|
91.016
|
0
|
COLO-800 | GDSC1000 |
5.261
|
N/A
|
1.25e+03
|
89.478
|
0
|
COLO-829 | GDSC1000 |
4.657
|
N/A
|
1e+06
|
90.687
|
0
|
MKL-2 | GDSC1000 |
7.693
|
258
|
258
|
0.000
|
0
|
CP67-MEL | GDSC1000 |
15.083
|
N/A
|
1e+06
|
69.833
|
0
|
LB373-MEL-D | GDSC1000 |
0.355
|
3.74
|
3.74
|
0.000
|
0
|
LB2518-MEL | GDSC1000 |
9.665
|
N/A
|
0.000186
|
80.670
|
0
|
CP66-MEL | GDSC1000 |
3.745
|
N/A
|
324
|
92.510
|
0
|
GAK | GDSC1000 |
8.084
|
N/A
|
1e+06
|
83.832
|
0
|
SK-MEL-2 | GDSC1000 |
3.998
|
N/A
|
0.153
|
91.667
|
0
|
MZ2-MEL | GDSC1000 |
6.230
|
N/A
|
161
|
87.539
|
0
|
A253 | GDSC1000 |
4.265
|
N/A
|
8.5e+05
|
90.259
|
0
|
HT-144 | GDSC1000 |
8.847
|
N/A
|
15.2
|
82.306
|
0
|
DJM-1 | GDSC1000 |
5.242
|
N/A
|
0.013
|
89.515
|
0
|
SH-4 | GDSC1000 |
10.224
|
N/A
|
13.7
|
79.553
|
0
|
SK-MEL-1 | GDSC1000 |
4.063
|
N/A
|
0.011
|
95.623
|
0
|
A388 | GDSC1000 |
6.611
|
73
|
73
|
0.000
|
0
|
A2058 | gCSI |
2.383
|
2.05
|
2.05
|
0.000
|
0
|
A375 | gCSI |
3.407
|
0.901
|
0.901
|
0.000
|
0.0221
|
A388 | gCSI |
28.217
|
1.69
|
1.69
|
0.000
|
0.259
|
A431 | gCSI |
0.432
|
1.57
|
1.57
|
0.000
|
0
|
C32 | gCSI |
4.737
|
1.3e+03
|
1.3e+03
|
0.000
|
0
|
CHL-1 | gCSI |
6.893
|
N/A
|
0.00349
|
89.082
|
0.00141
|
COLO-679 | gCSI |
4.650
|
N/A
|
0.0078
|
91.226
|
0
|
COLO-800 | gCSI |
7.074
|
N/A
|
0.0358
|
83.200
|
0.00432
|
COLO-829 | gCSI |
6.760
|
1.42
|
1.42
|
0.000
|
0
|
G-361 | gCSI |
8.489
|
7.51
|
7.51
|
0.000
|
0
|
HMV-II | gCSI |
9.858
|
8.43e+06
|
1e+06
|
10.974
|
0
|
Hs 294T | gCSI |
2.584
|
1.15
|
1.15
|
0.000
|
0
|
Hs 695T | gCSI |
3.128
|
N/A
|
0.491
|
71.341
|
0.0081
|
Hs 852.T | gCSI |
4.172
|
3.44
|
3.44
|
0.000
|
0
|
IGR-1 | gCSI |
3.658
|
0.965
|
0.965
|
0.000
|
0.0222
|
IGR-37 | gCSI |
4.845
|
6.97
|
6.97
|
0.000
|
0
|
IGR-39 | gCSI |
3.907
|
N/A
|
0.263
|
74.351
|
0.0201
|
IPC-298 | gCSI |
2.081
|
5.73
|
5.73
|
0.000
|
0
|
MEL-HO | gCSI |
10.364
|
567
|
567
|
0.000
|
0
|
MEL-JUSO | gCSI |
1.016
|
1.24
|
1.24
|
0.000
|
0
|
Mewo | gCSI |
9.914
|
153
|
153
|
0.000
|
0
|
RPMI-7951 | gCSI |
2.303
|
3.8
|
3.8
|
0.000
|
0
|
RVH-421 | gCSI |
3.218
|
5.79
|
5.79
|
0.000
|
0
|
SK-MEL-1 | gCSI |
2.569
|
1.44e+05
|
1.44e+05
|
0.000
|
0
|
SK-MEL-2 | gCSI |
5.816
|
N/A
|
0.00393
|
88.369
|
0
|
SK-MEL-24 | gCSI |
4.262
|
6.05
|
6.05
|
0.000
|
0
|
SK-MEL-3 | gCSI |
3.105
|
4.7
|
4.7
|
0.000
|
0
|
SK-MEL-30 | gCSI |
6.691
|
40.5
|
40.5
|
0.000
|
0
|
WM-115 | gCSI |
6.362
|
9.98e+04
|
9.98e+04
|
0.000
|
0
|
WM-266-4 | gCSI |
4.750
|
N/A
|
0.335
|
61.930
|
0.032
|
A375 | CTRPv2 |
25.195
|
4.75
|
4.73
|
0.581
|
0.239
|
MEL-HO | CTRPv2 |
25.007
|
4.88
|
4.88
|
0.113
|
0.241
|
SK-MEL-1 | CTRPv2 |
21.469
|
6.78
|
6.69
|
2.444
|
0.205
|
Hs 944.T | CTRPv2 |
23.800
|
5.79
|
5.79
|
0.000
|
0.21
|
MEL-JUSO | CTRPv2 |
22.859
|
6.14
|
6.14
|
0.000
|
0.212
|
SK-MEL-31 | CTRPv2 |
16.873
|
11.5
|
11.5
|
0.000
|
0.153
|
SK-MEL-5 | CTRPv2 |
17.059
|
11.2
|
11.2
|
0.000
|
0.162
|
IPC-298 | CTRPv2 |
19.723
|
8.49
|
8.49
|
0.000
|
0.185
|
SK-MEL-30 | CTRPv2 |
17.674
|
10.5
|
10.5
|
0.000
|
0.168
|
A375 | CTRPv2 |
17.264
|
11.1
|
11.1
|
0.000
|
0.155
|
WM1799 | CTRPv2 |
20.680
|
7.86
|
7.86
|
0.000
|
0.185
|
WM-793 | CTRPv2 |
18.553
|
9.79
|
9.79
|
0.000
|
0.165
|
G-361 | CTRPv2 |
20.310
|
7.82
|
7.58
|
2.810
|
0.184
|
Hs 852.T | CTRPv2 |
28.666
|
2.09
|
1.87
|
16.261
|
0.271
|
Hs 936.T | CTRPv2 |
18.215
|
14.3
|
14.3
|
0.000
|
0.14
|
COLO-800 | CTRPv2 |
17.671
|
5.45
|
5.26
|
6.556
|
0.166
|
K029AX | CTRPv2 |
19.174
|
5.13
|
5.13
|
0.000
|
0.182
|
COLO-829 | CTRPv2 |
26.323
|
4.45
|
4.45
|
0.000
|
0.233
|
IGR-1 | CTRPv2 |
28.356
|
3.02
|
2.94
|
5.162
|
0.273
|
SH-4 | CTRPv2 |
29.498
|
2.99
|
2.97
|
1.027
|
0.286
|
A253 | CTRPv2 |
8.476
|
29.3
|
29.3
|
0.000
|
0.0697
|
C32 | CTRPv2 |
19.509
|
8.99
|
8.99
|
0.000
|
0.172
|
HT-144 | CTRPv2 |
24.598
|
4.85
|
4.78
|
2.503
|
0.235
|
Hs 294T | CTRPv2 |
26.477
|
3.98
|
3.9
|
2.637
|
0.251
|
SK-MEL-2 | CTRPv2 |
12.747
|
17.5
|
17.5
|
0.000
|
0.119
|
A101D | CTRPv2 |
25.276
|
4.5
|
4.45
|
2.513
|
0.243
|
A2058 | CTRPv2 |
22.971
|
5.79
|
5.73
|
2.210
|
0.221
|
COLO-792 | CTRPv2 |
29.255
|
2.96
|
2.92
|
2.431
|
0.281
|
HMCB | CTRPv2 |
9.956
|
23.5
|
23.5
|
0.000
|
0.0909
|
IGR-39 | CTRPv2 |
14.034
|
N/A
|
3.38
|
50.855
|
0.118
|
Mewo | CTRPv2 |
22.115
|
6.64
|
6.38
|
2.653
|
0.196
|
WM-115 | CTRPv2 |
23.743
|
5.58
|
5.58
|
0.000
|
0.229
|
WM-266-4 | CTRPv2 |
23.183
|
5.66
|
5.6
|
2.227
|
0.223
|
Hs 895.T | CTRPv2 |
22.208
|
6.67
|
6.67
|
0.000
|
0.2
|
RVH-421 | CTRPv2 |
22.560
|
5.98
|
5.89
|
2.863
|
0.216
|
Hs 839.T | CTRPv2 |
12.214
|
18.7
|
18.7
|
0.000
|
0.111
|
WM-88 | CTRPv2 |
21.686
|
3.28
|
2.6
|
30.231
|
0.199
|
WM-983B | CTRPv2 |
22.002
|
5.79
|
4.68
|
13.878
|
0.195
|
CJM | CTRPv2 |
22.692
|
5.8
|
5.7
|
3.637
|
0.217
|
SK-MEL-3 | CTRPv2 |
23.787
|
5.5
|
5.48
|
0.532
|
0.229
|
IGR-37 | CTRPv2 |
18.572
|
9.56
|
9.56
|
0.000
|
0.177
|
Hs 934.T | CTRPv2 |
25.060
|
5.09
|
5.09
|
0.000
|
0.221
|
Hs 688(A).T | CTRPv2 |
25.668
|
4.69
|
4.69
|
0.000
|
0.23
|
Hs 940.T | CTRPv2 |
26.427
|
4.16
|
4.15
|
0.630
|
0.255
|
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