Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 1.287 9.44 9.44 0.000 0
BT-20 CCLE 8.592 N/A 0.0185 88.499 0.0082
BT-474 CCLE 0.653 11.5 11.5 0.000 0
BT-549 CCLE 2.682 7.39 7.39 0.000 0.0175
CAL-85-1 CCLE 2.360 9.96 9.96 0.000 0
CAMA-1 CCLE 0.877 11.1 10 17.500 0
EFM-19 CCLE 4.388 7.61 7.61 0.000 0.0269
HARA CCLE 0.768 12.3 10 27.812 0
HCC1187 CCLE 1.900 N/A 0.0052 96.200 0
HCC1395 CCLE 6.334 N/A 0.0113 92.212 0
HCC1569 CCLE 0.490 15.3 11 36.657 0
HCC1806 CCLE 5.474 6.9 6.9 0.000 0.0354
HCC1954 CCLE 2.024 8.16 8.16 0.000 0
HCC70 CCLE 1.480 9.04 9.04 0.000 0
HDQ-P1 CCLE 2.237 8.9 8.9 0.000 0
HMC-1-8 CCLE 4.060 7.08 7.08 0.000 0.0265
Hs-578-T CCLE 2.310 9.92 9.92 0.000 0
Hs 739.T CCLE 7.055 4.64 3.13 39.609 0.0562
MB 157 CCLE 1.850 8.41 8.41 0.000 0
MCF7 CCLE 9.017 3.92 3.92 0.000 0.0792
MDA-MB-157 CCLE 9.827 5.42e+04 5.42e+04 0.000 0
MDA-MB-175-VII CCLE 12.542 4.39e+11 1e+06 34.835 0
MDA-MB-415 CCLE 0.975 10.3 10.3 0.000 0
MDA-MB-436 CCLE 2.271 7.85 7.85 0.000 0.0138
MDA-MB-453 CCLE 4.670 N/A 3.46 55.496 0.0322
MDA-MB-468 CCLE 5.795 5.95 3.5 44.020 0.044
SK-BR-3 CCLE 0.238 N/A 3.81e-05 99.763 0
T47D CCLE 2.847 N/A 3.69 70.733 0.0145
UACC-812 CCLE 2.270 3.55e+03 3.55e+03 0.000 0
ZR-75-1 CCLE 10.422 N/A 5.14e+05 75.356 0
ZR-75-30 CCLE 3.225 N/A 0.0472 93.550 0
HCC2218 GDSC1000 8.310 N/A 1e-06 91.690 0
BT-474 GDSC1000 2.088 N/A 0.000509 97.912 0
HCC1599 GDSC1000 11.559 79.4 79.4 0.000 0
MRK-nu-1 GDSC1000 10.243 3.26e+03 2.46 48.928 0
EVSA-T GDSC1000 0.146 4.69 4.69 0.000 0
UACC-812 GDSC1000 0.138 N/A 3.95 52.028 0
DU-4475 GDSC1000 3.935 N/A 0.125 92.131 0
HCC1500 GDSC1000 10.099 N/A 0.0111 89.110 0.00773
HCC2157 GDSC1000 0.000 N/A 0.00781 100.000 0
HCC1187 GDSC1000 8.283 18 18 0.000 0
MDA-MB-134-VI GDSC1000 0.480 N/A 0.558 97.917 0
OCUB-M GDSC1000 3.197 110 110 0.000 0
CAL-148 GDSC1000 5.773 N/A 0.00499 94.164 0
MFM-223 GDSC1000 4.242 N/A 0.193 91.515 0
COLO-824 GDSC1000 0.875 N/A 0.604 98.249 0
AU565 gCSI 1.548 N/A 0.0755 96.904 0
BT-20 gCSI 1.051 2.62 2.62 0.000 0
BT-474 gCSI 0.979 N/A 0.000625 98.042 0
BT-549 gCSI 0.114 N/A 1.85 50.861 0
CAL-120 gCSI 4.195 N/A 0.00467 91.891 0
CAL-148 gCSI 4.228 663 663 0.000 0
CAL-51 gCSI 3.371 1.1 1.1 0.000 0
CAMA-1 gCSI 0.794 N/A 0.00252 98.835 0
EFM-19 gCSI 0.113 N/A 2.56 72.490 0
EVSA-T gCSI 2.020 N/A 0.00784 95.961 0
HCC1143 gCSI 1.418 N/A 0.366 87.670 0.00114
HCC1187 gCSI 0.272 2.34 1.55 40.516 0
HCC1419 gCSI 0.000 N/A 0.000153 100.000 0
HCC1806 gCSI 1.704 N/A 0.374 84.872 0.00342
HCC1937 gCSI 1.051 N/A 0.00378 97.897 0
HCC1954 gCSI 1.429 N/A 0.121 94.239 0
HCC2218 gCSI 10.589 7.93 7.93 0.000 0.0957
HCC38 gCSI 0.597 N/A 0.000185 99.383 0
HDQ-P1 gCSI 1.979 N/A 0.00687 96.041 0
Hs-578-T gCSI 0.032 N/A 1.96 82.972 0
MCF7 gCSI 3.052 N/A 0.383 72.193 0.016
MDA-MB-157 gCSI 1.968 N/A 0.362 83.066 0.00538
MDA-MB-175-VII gCSI 1.603 N/A 0.00106 96.794 0
MDA-MB-231 gCSI 3.075 N/A 0.338 75.162 0.0152
MDA-MB-436 gCSI 2.648 N/A 1e+06 75.990 0
MDA-MB-453 gCSI 1.437 198 198 0.000 0
MDA-MB-468 gCSI 0.900 N/A 1 70.938 0.000714
MFM-223 gCSI 3.103 33.3 33.3 0.000 0
SK-BR-3 gCSI 0.924 N/A 0.0135 98.153 0
T47D gCSI 1.138 N/A 0.181 94.150 0
600MPE GRAY 21.973 2.05 2.05 0.000 0.195
AU565 GRAY 12.709 6.49 6.42 1.243 0.115
AU565 GRAY 13.474 6.64 6.64 0.000 0.112
BT-20 GRAY 11.396 7.95 7.95 0.000 0.0994
BT-474 GRAY 8.686 11 11 0.000 0.078
BT-549 GRAY 15.299 4.79 4.79 0.000 0.135
CAMA-1 GRAY 9.354 10.2 10.2 0.000 0.083
HCC1143 GRAY 19.177 3.13 3.13 0.000 0.163
HCC1143 GRAY 13.205 6.44 6.44 0.000 0.114
HCC1187 GRAY 17.460 4.18 4.18 0.000 0.144
HCC1395 GRAY 9.581 9.87 9.87 0.000 0.0849
HCC1419 GRAY 5.044 17.7 17.7 0.000 0.0436
HCC1428 GRAY 9.424 10 10 0.000 0.0842
HCC1428 GRAY 8.237 11.6 11.6 0.000 0.074
HCC1569 GRAY 19.081 2.87 2.84 0.818 0.173
HCC1569 GRAY 18.363 3.18 3.18 0.000 0.166
HCC1806 GRAY 23.863 1.43 1.31 5.467 0.216
HCC1937 GRAY 12.989 6.04 5.95 2.911 0.123
HCC1937 GRAY 10.413 8.81 8.81 0.000 0.0936
HCC3153 GRAY 8.768 10.9 10.9 0.000 0.0782
HCC70 GRAY 13.729 5.98 5.98 0.000 0.119
Hs-578-T GRAY 21.454 1.99 1.89 3.941 0.196
MCF10A GRAY 19.398 2.8 2.8 0.000 0.174
MCF12A GRAY 14.308 5.47 5.47 0.000 0.126
MCF7 GRAY 21.679 2.04 2.03 0.339 0.2
MDA-MB-134-VI GRAY 17.761 3.55 3.55 0.000 0.155
MDA-MB-157 GRAY 16.279 4.18 4.18 0.000 0.146
MDA-MB-231 GRAY 17.271 3.81 3.81 0.000 0.15
MDA-MB-361 GRAY 10.095 9.34 9.34 0.000 0.0883
MX-1 GRAY 16.391 4.21 4.21 0.000 0.144
SK-BR-3 GRAY 9.146 10.4 10.4 0.000 0.0821
SUM 1315M02 GRAY 11.589 7.3 7.21 2.524 0.109
SUM 1315M02 GRAY 10.675 8.28 8.2 2.037 0.0995
SUM 149PT GRAY 16.948 3.75 3.7 1.159 0.154
SUM 159PT GRAY 22.802 1.72 1.68 1.790 0.21
SUM185PE GRAY 10.414 8.88 8.88 0.000 0.0923
SUM 229PE GRAY 18.000 3.17 3.1 2.416 0.167
SUM 229PE GRAY 17.933 3.23 3.18 1.800 0.167
T47D GRAY 11.072 8.42 8.42 0.000 0.095
T47D_KBluc GRAY 10.302 9.02 9.02 0.000 0.091
UACC-812 GRAY 7.232 13.3 13.3 0.000 0.0644
ZR-75-1 GRAY 14.708 6.06 6.06 0.000 0.119
ZR75B GRAY 17.511 3.82 3.82 0.000 0.149
21MT1 GRAY 9.606 9.83 9.83 0.000 0.0853
21NT GRAY 10.212 9.09 9.09 0.000 0.0908
HCC1187 GRAY 22.498 1.87 1.64 5.801 0.195
HCC1954 GRAY 15.786 4.58 4.58 0.000 0.138
HCC38 GRAY 17.539 3.95 3.95 0.000 0.147
LY2 GRAY 20.971 2.17 2.13 1.933 0.196
MCF10F GRAY 18.455 3.17 3.17 0.000 0.165
MDA-MB-175-VII GRAY 9.219 10.3 10.3 0.000 0.0824
MDA-MB-453 GRAY 15.325 5.08 5.08 0.000 0.13
SUM 52PE GRAY 25.214 1.4 1.4 0.000 0.22
184A1 GRAY 15.498 5.32 5.32 0.000 0.127
184B5 GRAY 14.156 5.86 5.86 0.000 0.12
21MT1 GRAY 11.999 7.39 7.39 0.000 0.104
21MT1 GRAY 13.622 6.2 6.2 0.000 0.116
HCC2185 GRAY 7.528 12.7 12.7 0.000 0.0676
MDA-MB-415 GRAY 14.465 5.58 5.58 0.000 0.123
SUM225CWN GRAY 3.946 23.2 23.2 0.000 0.029
BT-474 FIMM 11.862 3.54 3.54 0.000 0.1
BT-549 FIMM 3.310 8.07 8.07 0.000 0.0242
CAL-120 FIMM 15.144 2.64 2.64 0.000 0.128
HCC1143 FIMM 6.248 8.17 8.17 0.000 0.0406
HCC1599 FIMM 3.033 13.3 10.1 20.572 0
HCC1937 FIMM 13.927 2.89 2.89 0.000 0.12
Hs-578-T FIMM 3.039 8.42 8.42 0.000 0.0215
MCF7 FIMM 34.192 1.09 1.09 0.000 0.269
MDA-MB-231 FIMM 22.165 1.37 1.37 0.000 0.192
MDA-MB-436 FIMM 43.522 0.207 0.207 0.000 0.375
MDA-MB-468 FIMM 11.400 3.64 3.64 0.000 0.0977
MFM-223 FIMM 26.455 4.46 4.46 0.000 0.185
SK-BR-3 FIMM 7.722 4.98 4.98 0.000 0.0676
T47D FIMM 11.899 4.37 4.37 0.000 0.0892
ZR-75-1 FIMM 9.864 0.00507 0.00507 0.000 0.0736
CAL-148 FIMM 5.458 9.6 9.31 2.188 0.033
CAL-51 FIMM 3.206 8.18 8.18 0.000 0.0233
CAL-85-1 FIMM 10.623 6.47 6.47 0.000 0.071
DU-4475 FIMM 5.933 5.96 5.94 0.752 0.0499
HDQ-P1 FIMM 8.683 7.03 7.03 0.000 0.058
MDA-MB-453 FIMM 10.160 4.78 4.78 0.000 0.0774
KPL-1 CTRPv2 21.539 7 7 0.146 0.207
CAL-120 CTRPv2 15.777 12.7 12.7 0.380 0.149
HDQ-P1 CTRPv2 13.699 16.2 16.2 0.000 0.121
JIMT-1 CTRPv2 16.010 12.1 12 2.393 0.151
HARA CTRPv2 29.252 3.14 3.05 1.722 0.263
CAMA-1 CTRPv2 16.675 11.6 11.6 0.437 0.158
MCF7 CTRPv2 32.959 2.25 2.25 0.000 0.292
HCC1806 CTRPv2 19.773 8.51 8.51 0.000 0.18
HCC1954 CTRPv2 21.900 6.77 6.77 0.000 0.205
HMC-1-8 CTRPv2 32.102 2.36 2.36 0.000 0.296
HCC1937 CTRPv2 15.543 13.1 13.1 0.000 0.143
CAL-148 CTRPv2 30.629 2.86 2.86 0.000 0.271
CAL-51 CTRPv2 34.229 1.95 1.95 0.000 0.305
HCC1395 CTRPv2 22.273 6.58 6.58 0.000 0.203
CAL-51 CTRPv2 33.700 2.08 2.08 0.000 0.298
MDA-MB-231 CTRPv2 21.883 7.01 7.01 0.000 0.194
HCC1143 CTRPv2 25.997 4.74 4.74 0.000 0.226
ZR-75-1 CTRPv2 21.170 7.5 7.5 0.000 0.188
HCC1428 CTRPv2 12.252 9.71 9.47 4.835 0.113
HCC38 CTRPv2 13.126 10.7 10.7 0.000 0.105
BT-549 CTRPv2 13.093 9.19 8.77 5.316 0.115
HCC202 CTRPv2 5.679 22.8 22.8 0.000 0.0411
DU-4475 CTRPv2 29.658 2.45 2.24 8.787 0.278
HCC1500 CTRPv2 24.355 4.81 4.43 6.436 0.221
Hs-578-T CTRPv2 32.295 2.28 2.25 0.713 0.297
MDA-MB-468 CTRPv2 29.021 2.99 2.94 2.903 0.28
CAL-85-1 CTRPv2 21.475 5.31 4.88 14.193 0.203
BT-20 CTRPv2 9.229 25.4 25.4 0.000 0.0837
HCC1419 CTRPv2 12.832 15.1 13.9 14.245 0.118
ZR-75-30 CTRPv2 6.464 34.5 29 20.801 0.0525
EFM-192A CTRPv2 11.917 11.5 11.5 0.000 0.0971
MDA-MB-157 CTRPv2 12.301 6.72 4.46 40.327 0.106
MDA-MB-361 CTRPv2 12.774 18.3 18.3 0.000 0.11
T47D CTRPv2 14.542 14.9 14.9 0.000 0.128
BT-474 CTRPv2 14.183 15.1 15 0.342 0.133
HCC2218 CTRPv2 14.782 13.9 13.8 1.710 0.139
SK-BR-3 CTRPv2 15.782 12.1 11.8 4.435 0.148
MDA-MB-453 CTRPv2 18.123 9.92 9.89 0.662 0.172
AU565 CTRPv2 23.488 5.85 5.85 0.000 0.211
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