Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MFM-223 GDSC1000 3.174 N/A 1.4 65.936 0.0101
MDA-MB-231 GDSC1000 2.069 N/A 0.74 88.514 0.000851
UACC-893 GDSC1000 7.037 N/A 0.165 84.477 0.0121
HCC1937 GDSC1000 17.951 2.83 2.83 0.000 0
CAL-51 GDSC1000 0.329 N/A 6.37e-05 99.671 0
Hs-578-T GDSC1000 2.186 N/A 1.05 82.078 0.0039
EFM-19 GDSC1000 5.156 N/A 0.356 83.438 0.0171
HARA GDSC1000 22.291 0.449 0.213 44.849 0.186
HCC70 GDSC1000 2.222 N/A 248 95.556 0
HDQ-P1 GDSC1000 9.097 N/A 0.336 71.731 0.0545
BT-20 GDSC1000 9.127 N/A 1e+06 67.448 0
HCC1954 GDSC1000 6.663 N/A 0.431 75.926 0.0351
MRK-nu-1 GDSC1000 1.144 N/A 1.24 97.713 0
MCF7 GDSC1000 2.359 N/A 0.111 95.473 0
BT-483 GDSC1000 0.351 3.75 3.75 0.000 0
HCC1187 GDSC1000 10.206 N/A 0.0261 84.536 0.0132
EVSA-T GDSC1000 1.202 N/A 0.138 97.506 0
MDA-MB-468 GDSC1000 4.784 4.96 1.62 44.268 0.0217
HCC1419 GDSC1000 3.287 N/A 250 93.427 0
HCC2218 GDSC1000 3.637 N/A 17 70.504 0
HCC38 GDSC1000 0.025 N/A 0.0164 99.969 0
CAL-120 GDSC1000 3.641 N/A 0.334 88.712 0.00261
T47D GDSC1000 5.418 N/A 1e+06 89.165 0
MDA-MB-415 GDSC1000 0.000 N/A 0.00781 100.000 0
MDA-MB-175-VII GDSC1000 2.749 N/A 1.44 60.875 0.0128
HCC1500 GDSC1000 5.893 N/A 0.453 79.980 0.0111
OCUB-M GDSC1000 0.822 2.99 2.99 0.000 0
JIMT-1 GDSC1000 13.292 1.76 0.642 40.037 0.0911
HCC2157 GDSC1000 2.154 N/A 0.743 87.991 0.00138
EFM-192A GDSC1000 4.061 N/A 1.42 70.066 0.00723
HCC1395 GDSC1000 7.275 N/A 0.177 83.377 0.0266
HCC1143 GDSC1000 2.879 N/A 0.584 87.052 0.00384
HCC202 GDSC1000 0.000 N/A 0.00781 100.000 0
MDA-MB-361 GDSC1000 3.067 2.01 2.01 0.000 0
ZR-75-30 GDSC1000 3.662 N/A 0.995 71.517 0.0175
MDA-MB-330 GDSC1000 3.552 N/A 1.78 85.346 0.00353
MDA-MB-453 GDSC1000 0.698 3.13 3.13 0.000 0
COLO-824 GDSC1000 0.000 N/A 0.00802 100.000 0
BT-549 GDSC1000 17.844 N/A 0.127 64.218 0.0894
HCC1569 GDSC1000 2.951 N/A 1.55e+04 94.098 0
MDA-MB-436 GDSC1000 4.400 N/A 0.664 77.945 0.0192
DU-4475 GDSC1000 3.024 5.53 5.53 0.000 0
BT-474 GDSC1000 1.498 N/A 0.304 95.593 0
AU565 GDSC1000 0.918 2.9 2.9 0.000 0
HCC1428 GDSC1000 3.394 N/A 1.91 79.435 5.47e-05
CAL-85-1 GDSC1000 1.254 N/A 0.268 96.539 0
AU565 GRAY 25.790 3.71 3.71 0.000 0.232
BT-474 GRAY 9.891 N/A 4.24 59.713 0.0777
CAMA-1 GRAY 13.329 N/A 3.13 50.531 0.103
HCC1143 GRAY 18.439 11.3 6.2 18.675 0.147
HCC1419 GRAY 13.319 30.2 14.2 22.242 0.0981
HCC1806 GRAY 26.480 2.41 2.04 12.421 0.245
HCC2185 GRAY 7.448 N/A 5.49 66.959 0.0533
MCF10F GRAY 20.948 3.16 1.35 37.348 0.181
BT-20 GRAY 27.553 1.85 1.38 17.192 0.251
BT-483 GRAY 12.433 10.5 4.54 48.237 0.106
ZR-75-1 GRAY 7.137 40.3 40.3 0.000 0.0637
CAMA-1 GRAY 9.496 N/A 379 51.562 0
HCC1187 GRAY 21.141 5.67 4.21 14.668 0.185
HCC1428 GRAY 20.680 7.08 7.08 0.000 0.188
HCC1569 GRAY 25.233 2.36 1.74 19.839 0.23
HCC1937 GRAY 24.321 2.36 1.67 23.468 0.221
HCC1954 GRAY 29.736 2.29 2.29 0.000 0.264
HCC2185 GRAY 9.086 139 14.2 44.319 0.0604
HCC3153 GRAY 8.016 N/A 8.28 59.152 0.0518
HCC3153 GRAY 21.971 5.57 5.42 3.011 0.206
HCC38 GRAY 34.447 0.978 0.938 5.003 0.332
Hs-578-T GRAY 31.383 1.71 1.68 1.161 0.293
MCF10A GRAY 29.468 1.46 1.22 13.930 0.275
MCF7 GRAY 17.060 71 1.81 46.307 0.124
MDA-MB-134-VI GRAY 10.636 N/A 0.000368 78.728 0
MX-1 GRAY 27.799 2.85 2.85 0.000 0.252
SUM 149PT GRAY 37.713 0.788 0.788 0.000 0.347
SUM 149PT GRAY 34.385 1.17 1.14 1.197 0.316
SUM 52PE GRAY 22.919 6.31 1.92 27.215 0.183
SUM 52PE GRAY 26.516 2.85 2.57 6.826 0.244
UACC-812 GRAY 12.881 1.33e+03 3.68 49.965 0.0971
UACC-812 GRAY 20.557 453 453 0.000 0
ZR-75-1 GRAY 17.982 9.6 9.39 2.248 0.166
ZR75B GRAY 13.941 14.6 7.76 30.213 0.116
184A1 GRAY 21.164 0.892 0.392 38.655 0.184
184B5 GRAY 23.201 1.15 0.741 21.613 0.205
HCC70 GRAY 22.800 1.46 1.31 9.323 0.211
MB 157 GRAY 36.410 0.287 0.259 3.888 0.328
MDA-MB-157 GRAY 20.709 1.68 1.56 12.810 0.197
MDA-MB-231 GRAY 18.866 2.33 2.19 10.732 0.179
MDA-MB-453 GRAY 13.543 3.4 2.68 30.824 0.123
600MPE GRAY 6.957 N/A 5.93 68.318 0.0441
BT-474 GRAY 20.915 5.35 2.96 23.878 0.179
HCC1395 GRAY 28.545 2.19 2 6.113 0.264
HCC1395 GRAY 27.084 2.64 2.48 5.664 0.255
MDA-MB-134-VI GRAY 2.726 N/A 21 77.528 0.0135
MDA-MB-175-VII GRAY 21.649 4.32 2.3 26.338 0.187
MDA-MB-231 GRAY 33.542 1.17 1.08 4.751 0.31
MX-1 GRAY 19.267 17.9 17.9 0.000 0.141
SUM185PE GRAY 7.287 N/A 3.17 72.806 0.0473
SUM225CWN GRAY 20.345 5.25 2.71 27.621 0.174
BT-20 GRAY 24.814 3.03 2.56 12.804 0.229
BT-483 GRAY 8.279 N/A 6.72 60.586 0.0581
HCC1428 GRAY 17.639 11.6 11.6 0.000 0.148
HCC38 GRAY 33.476 1.19 1.16 3.234 0.324
HCC70 GRAY 28.625 2.35 2.15 4.475 0.258
LY2 GRAY 23.883 3.9 3.4 9.183 0.218
MCF12A GRAY 31.745 1.44 1.26 6.690 0.29
MDA-MB-175-VII GRAY 19.553 9.55 9.55 0.000 0.163
MDA-MB-175-VII GRAY 15.917 39.4 2.42 45.597 0.119
MDA-MB-361 GRAY 15.803 29.6 1.75 49.697 0.129
MDA-MB-361 GRAY 14.885 40.7 2.78 46.850 0.113
MDA-MB-415 GRAY 22.303 5.93 5.93 0.000 0.197
MX-1 GRAY 20.252 8.05 5.84 11.655 0.168
SK-BR-3 GRAY 22.294 5.84 5.84 0.000 0.199
SUM 1315M02 GRAY 30.998 1.4 1.12 11.211 0.282
SUM 159PT GRAY 33.407 1.38 1.38 0.000 0.305
SUM225CWN GRAY 22.823 31.8 19.2 6.906 0.156
SUM 229PE GRAY 29.946 1.9 1.64 6.698 0.269
T47D GRAY 20.607 6.43 6.24 4.336 0.196
UACC-812 GRAY 18.402 6.51 2.17 38.203 0.153
BT-474 GRAY 12.866 5.54 1.66 44.839 0.105
BT-549 GRAY 25.582 1.28 1.28 0.000 0.229
HCC1569 GRAY 14.006 3.35 1.91 36.877 0.121
Hs-578-T GRAY 14.747 3.61 3.2 18.931 0.137
LY2 GRAY 11.591 4.18 2.83 39.481 0.102
MCF12A GRAY 23.551 1.46 1.37 5.065 0.217
MDA-MB-361 GRAY 14.479 2.4 1.71 37.236 0.129
MDA-MB-415 GRAY 7.026 N/A 1.79 69.065 0.0486
SUM 1315M02 GRAY 16.359 1.98 1.54 31.426 0.149
T47D_KBluc GRAY 3.923 N/A 2.98 79.063 0.0196
Hs-578-T FIMM 6.540 6.35 6.35 0.000 0.049
KPL-1 CTRPv2 18.749 9.4 9.4 0.000 0.174
CAL-120 CTRPv2 19.876 8.47 8.47 0.000 0.179
HDQ-P1 CTRPv2 35.669 1.71 1.71 0.000 0.315
JIMT-1 CTRPv2 17.512 6.14 5.93 2.861 0.153
HARA CTRPv2 31.901 2.37 2.31 1.541 0.289
CAMA-1 CTRPv2 14.013 4.35e+03 4.35e+03 0.000 0
MCF7 CTRPv2 7.173 N/A 2.41 77.466 0.0378
HCC1806 CTRPv2 28.631 3.47 3.47 0.000 0.255
HCC1954 CTRPv2 34.270 1.92 1.92 0.000 0.308
HMC-1-8 CTRPv2 6.046 10.1 10.1 0.000 0.0508
HCC1937 CTRPv2 22.508 6.49 6.49 0.000 0.202
CAL-148 CTRPv2 20.931 3.21 2.41 34.214 0.19
CAL-51 CTRPv2 19.993 4.6 2.81 34.070 0.176
HCC1395 CTRPv2 20.741 3.77 2.69 32.590 0.187
CAL-51 CTRPv2 24.383 5.3 5.3 0.000 0.221
MDA-MB-231 CTRPv2 18.638 9.81 9.81 0.000 0.164
HCC1143 CTRPv2 18.120 5.86 5.86 0.000 0.159
ZR-75-1 CTRPv2 5.728 N/A 5.89 75.338 0.0334
HCC1428 CTRPv2 18.833 9.42 9.42 0.000 0.17
HCC38 CTRPv2 22.230 5.54 4.93 10.942 0.203
BT-549 CTRPv2 16.365 5.62 3.06 44.535 0.141
HCC202 CTRPv2 20.130 7.41 1.37 45.934 0.164
DU-4475 CTRPv2 27.638 3.61 3.59 1.256 0.267
HCC1500 CTRPv2 20.614 6.76 6.25 9.029 0.191
Hs-578-T CTRPv2 24.343 4.84 4.69 4.186 0.231
MDA-MB-468 CTRPv2 26.393 4.29 4.29 0.000 0.24
CAL-85-1 CTRPv2 31.769 2.64 2.64 0.000 0.276
BT-20 CTRPv2 17.672 10.1 8.81 9.716 0.154
HCC1419 CTRPv2 23.383 7.54 7.54 0.000 0.189
ZR-75-30 CTRPv2 23.867 4.94 4.38 8.710 0.215
EFM-192A CTRPv2 20.105 8.8 8.8 0.000 0.172
MDA-MB-157 CTRPv2 33.323 4.22 4.22 0.000 0.262
MDA-MB-361 CTRPv2 16.715 12.5 12.5 0.000 0.142
T47D CTRPv2 21.750 6.17 5.98 5.757 0.208
BT-474 CTRPv2 36.279 1.55 1.55 0.000 0.328
HCC2218 CTRPv2 25.338 4.65 4.49 2.473 0.229
SK-BR-3 CTRPv2 23.921 5.04 4.93 4.055 0.23
MDA-MB-453 CTRPv2 23.688 4.92 4.75 6.377 0.226
AU565 CTRPv2 25.944 3.8 3.65 6.782 0.248
MDA-MB-415 CTRPv2 17.611 10.9 10.9 0.000 0.155
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