Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MMAC-SF GDSC1000 79.554 0.000196 0.000188 3.453 0.773
A101D GDSC1000 79.765 0.000213 0.00021 1.320 0.775
IST-MEL1 GDSC1000 53.814 0.000952 0.000941 2.387 0.521
CP66-MEL GDSC1000 63.025 0.00055 0.000542 3.161 0.612
A388 GDSC1000 68.562 0.000446 0.000446 0.000 0.666
COLO-829 GDSC1000 57.164 0.000722 0.000688 5.908 0.543
MZ2-MEL GDSC1000 66.551 0.000488 0.000485 0.534 0.637
A253 GDSC1000 53.329 0.00101 0.001 1.153 0.512
MKL-2 GDSC1000 33.049 0.00296 0.00288 5.507 0.312
DJM-1 GDSC1000 36.483 0.00268 0.00268 0.000 0.329
SK-MEL-2 GDSC1000 7.576 1.88 1.88 0.000 0
LB373-MEL-D GDSC1000 59.664 0.00069 0.000675 2.201 0.564
LB2518-MEL GDSC1000 66.528 0.000492 0.00049 0.515 0.649
COLO-800 GDSC1000 22.524 0.0204 0.0204 0.000 0
MKL-1-subclone-2 GDSC1000 28.652 0.00415 0.00415 0.000 0.257
MZ7-mel GDSC1000 50.267 0.00103 0.00095 8.504 0.47
SH-4 GDSC1000 82.781 0.00017 0.000169 0.138 0.809
HT-144 GDSC1000 68.209 0.000422 0.000415 2.306 0.658
SK-MEL-1 GDSC1000 8.349 N/A 0.00564 63.927 0.0499
A2058 gCSI 43.421 0.0219 0.0218 0.267 0.423
A375 gCSI 43.887 0.0212 0.0212 0.000 0.429
A431 gCSI 49.909 0.0123 0.0123 0.292 0.489
C32 gCSI 36.822 0.0382 0.038 1.065 0.357
CHL-1 gCSI 33.305 0.0494 0.0475 4.032 0.312
COLO-679 gCSI 37.816 0.036 0.036 0.051 0.368
COLO-800 gCSI 38.580 0.0329 0.0327 0.903 0.372
COLO-829 gCSI 37.671 0.0349 0.0343 1.906 0.357
G-361 gCSI 48.571 0.014 0.014 0.000 0.475
HMV-II gCSI 32.976 0.037 0.0316 16.107 0.307
Hs 294T gCSI 39.582 0.0305 0.0304 0.437 0.385
Hs 695T gCSI 37.373 0.0296 0.0284 7.824 0.36
Hs 852.T gCSI 14.765 0.274 0.274 0.000 0.137
IGR-1 gCSI 36.018 0.0422 0.0422 0.000 0.35
IGR-37 gCSI 36.541 0.0399 0.0398 0.456 0.355
IGR-39 gCSI 34.715 0.0464 0.0462 0.795 0.337
IPC-298 gCSI 44.469 0.0199 0.0199 0.295 0.432
MEL-HO gCSI 47.937 0.0148 0.0148 0.000 0.469
MEL-JUSO gCSI 35.978 0.042 0.042 0.326 0.347
Mewo gCSI 33.276 0.0525 0.0521 1.040 0.32
RPMI-7951 gCSI 41.938 0.0251 0.0251 0.000 0.409
RVH-421 gCSI 36.155 0.0415 0.0414 0.220 0.351
SK-MEL-1 gCSI 6.853 0.577 0.345 43.570 0.0544
SK-MEL-2 gCSI 37.002 0.0313 0.0302 7.155 0.357
SK-MEL-24 gCSI 24.024 0.11 0.101 8.079 0.219
SK-MEL-3 gCSI 33.036 0.043 0.04 9.823 0.313
SK-MEL-30 gCSI 40.964 0.0272 0.0271 0.225 0.399
WM-115 gCSI 32.509 0.0534 0.0526 3.053 0.314
WM-266-4 gCSI 23.952 0.117 0.115 2.886 0.223
RPMI-7951 CTRPv2 25.307 0.00847 0.00802 5.845 0.237
A375 CTRPv2 15.020 0.0272 0.0271 0.733 0.141
MEL-HO CTRPv2 26.001 0.00843 0.00833 1.917 0.249
SK-MEL-1 CTRPv2 9.385 0.0722 0.0722 0.000 0.0662
Hs 944.T CTRPv2 17.421 0.0207 0.0199 4.008 0.159
MEL-JUSO CTRPv2 18.177 0.0192 0.0189 2.521 0.168
SK-MEL-31 CTRPv2 15.102 0.0167 0.0153 8.533 0.131
SK-MEL-5 CTRPv2 21.499 0.00799 0.00752 10.867 0.202
IPC-298 CTRPv2 22.704 0.00798 0.0078 4.259 0.216
SK-MEL-30 CTRPv2 13.358 0.0203 0.0203 0.000 0.117
A375 CTRPv2 2.658 0.0586 0.0586 0.000 0.018
WM1799 CTRPv2 21.722 0.00893 0.00871 3.465 0.202
WM-793 CTRPv2 21.197 0.00947 0.00928 2.796 0.197
G-361 CTRPv2 16.697 0.0213 0.0213 0.000 0.125
Hs 852.T CTRPv2 4.290 0.0476 0.0476 0.000 0.0336
Hs 936.T CTRPv2 4.066 0.0494 0.0494 0.000 0.031
COLO-800 CTRPv2 27.515 0.00712 0.00692 2.836 0.257
K029AX CTRPv2 31.227 0.005 0.00498 0.783 0.303
COLO-829 CTRPv2 27.573 0.00797 0.00797 0.000 0.241
IGR-1 CTRPv2 18.121 0.0186 0.0179 5.230 0.168
SH-4 CTRPv2 32.128 0.00646 0.00618 5.042 0.303
A253 CTRPv2 26.321 0.00768 0.00717 5.933 0.243
C32 CTRPv2 26.370 0.00727 0.00703 6.337 0.253
HT-144 CTRPv2 25.494 0.00677 0.00613 13.500 0.24
Hs 294T CTRPv2 32.659 0.00401 0.00394 3.170 0.317
SK-MEL-2 CTRPv2 25.748 0.00665 0.00619 12.342 0.245
A101D CTRPv2 30.964 0.0052 0.00519 0.384 0.295
A2058 CTRPv2 16.761 0.0225 0.0223 1.384 0.159
COLO-792 CTRPv2 32.106 0.00469 0.00469 0.000 0.297
HMCB CTRPv2 25.473 0.00838 0.00802 5.239 0.239
IGR-39 CTRPv2 22.548 0.0114 0.01 9.136 0.202
Mewo CTRPv2 24.218 0.00904 0.00865 7.368 0.231
WM-115 CTRPv2 32.421 0.00377 0.00365 5.938 0.313
WM-266-4 CTRPv2 22.845 0.0115 0.0109 4.520 0.21
Hs 895.T CTRPv2 12.040 0.0326 0.0273 20.137 0.106
RVH-421 CTRPv2 27.311 0.00738 0.0073 1.703 0.262
Hs 839.T CTRPv2 8.137 N/A 8.35e-06 91.250 0
WM-88 CTRPv2 28.505 0.00615 0.00584 4.839 0.266
WM-983B CTRPv2 20.556 0.0145 0.0141 4.251 0.192
CJM CTRPv2 20.514 0.0156 0.0156 0.000 0.189
SK-MEL-3 CTRPv2 16.386 0.0148 0.00842 37.954 0.141
IGR-37 CTRPv2 21.945 0.0125 0.0123 3.301 0.21
Hs 688(A).T CTRPv2 1.554 N/A 0.0171 92.047 0
Hs 940.T CTRPv2 15.142 0.0303 0.0303 0.000 0.125
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