Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
A375 CTRPv2 1.869 32.5 32.5 0.000 0.0113
MEL-HO CTRPv2 3.274 N/A 4.27 87.553 0.0055
SK-MEL-1 CTRPv2 3.755 47.4 47.4 0.000 0.0295
Hs 944.T CTRPv2 26.935 4.26 4.26 0.000 0.235
MEL-JUSO CTRPv2 15.925 12.6 12.6 0.000 0.147
SK-MEL-31 CTRPv2 14.427 15.5 15.5 0.000 0.124
SK-MEL-5 CTRPv2 31.488 2.52 2.52 0.000 0.289
IPC-298 CTRPv2 10.615 21.9 21.9 0.000 0.0975
SK-MEL-30 CTRPv2 17.167 11.1 11.1 0.000 0.163
A375 CTRPv2 26.522 3.78 3.2 9.422 0.235
WM1799 CTRPv2 27.784 3.6 3.57 0.887 0.263
WM-793 CTRPv2 23.229 5.78 5.75 0.978 0.223
G-361 CTRPv2 31.978 2.3 2.28 1.129 0.304
Hs 852.T CTRPv2 44.358 0.663 0.663 0.000 0.404
Hs 936.T CTRPv2 16.971 11.6 11.6 0.000 0.15
COLO-800 CTRPv2 16.657 11.4 11.3 2.147 0.154
K029AX CTRPv2 15.561 13.5 13.5 0.000 0.136
COLO-829 CTRPv2 12.995 16.6 15.9 5.591 0.117
IGR-1 CTRPv2 10.635 21.3 20.8 4.242 0.0973
SH-4 CTRPv2 29.845 4.29 4.29 0.000 0.24
C32 CTRPv2 11.039 19.5 16.9 16.259 0.0962
HT-144 CTRPv2 7.522 33.2 33.2 0.000 0.0602
Hs 294T CTRPv2 8.941 27.8 27.8 0.000 0.0741
SK-MEL-2 CTRPv2 3.627 48.2 48.2 0.000 0.0283
A101D CTRPv2 4.403 2.12e+06 1e+06 7.436 0
A2058 CTRPv2 1.128 N/A 8.44 94.478 0
COLO-792 CTRPv2 19.748 4.71 4.64 2.312 0.185
HMCB CTRPv2 1.130 38.3 38.3 0.000 0
IGR-39 CTRPv2 15.059 7.93 5.83 35.444 0.134
Mewo CTRPv2 4.006 45.8 45.8 0.000 0.0319
WM-115 CTRPv2 19.740 8.12 7.98 2.812 0.186
WM-266-4 CTRPv2 13.816 15.9 15.9 0.000 0.124
Hs 895.T CTRPv2 0.842 82 82 0.000 0
SK-MEL-24 CTRPv2 5.451 38.5 38.5 0.000 0.0461
RVH-421 CTRPv2 4.111 45.2 45.2 0.000 0.033
Hs 839.T CTRPv2 3.978 46 46 -0.000 0.0317
WM-88 CTRPv2 26.719 3.63 3.54 4.977 0.257
WM-983B CTRPv2 5.184 39.7 39.7 0.000 0.0435
CJM CTRPv2 3.824 46.9 46.9 0.000 0.0302
SK-MEL-3 CTRPv2 19.844 7.86 7.57 4.723 0.184
IGR-37 CTRPv2 12.422 18.2 18.2 0.000 0.116
Hs 934.T CTRPv2 12.099 18.8 18.8 0.000 0.112
Hs 688(A).T CTRPv2 9.107 25.6 25.5 1.041 0.0824
Hs 940.T CTRPv2 22.195 6.55 6.55 0.045 0.213
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