Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
BT-474 GDSC1000 42.894 0.0461 0.024 20.267 0.366
HCC2218 GDSC1000 31.830 0.116 0.0772 27.422 0.29
HCC2218 GDSC1000 43.617 0.0277 0.0221 22.495 0.399
MFM-223 GDSC1000 0.000 N/A 0.00198 100.000 0
HCC1419 GDSC1000 16.505 2.07 0.357 45.220 0.13
HCC1419 GDSC1000 20.899 N/A 0.0429 52.847 0.161
MDA-MB-231 GDSC1000 1.682 N/A 2.54 86.386 0.003
MDA-MB-231 GDSC1000 5.095 N/A 0.00998 92.782 0
UACC-893 GDSC1000 34.210 0.106 0.0676 13.667 0.271
T47D GDSC1000 8.084 N/A 0.0764 76.158 0.0404
HCC1937 GDSC1000 4.739 5.47e+03 5.47e+03 0.000 0
HCC1937 GDSC1000 8.270 N/A 0.0233 85.044 0.0229
Hs-578-T GDSC1000 1.523 N/A 0.066 96.252 0
HDQ-P1 GDSC1000 7.574 N/A 0.382 74.331 0.0389
EFM-19 GDSC1000 9.026 7.65e+10 1e+06 35.350 0
EFM-19 GDSC1000 3.227 N/A 86 93.546 0
HARA GDSC1000 13.071 N/A 0.143 65.922 0.0837
HARA GDSC1000 23.182 2.92 1.74 6.900 0
CAMA-1 GDSC1000 2.001 N/A 2.66 85.146 0.000823
Hs-578-T GDSC1000 7.933 N/A 0.0232 84.134 0
HCC70 GDSC1000 7.728 N/A 0.053 83.641 0.0299
HCC70 GDSC1000 10.346 N/A 0.000181 87.526 0.00655
MB 157 GDSC1000 20.722 N/A 0.0789 52.835 0.147
UACC-893 GDSC1000 26.442 0.194 0.132 32.209 0.24
BT-20 GDSC1000 7.906 N/A 0.42 72.388 0.0443
BT-20 GDSC1000 22.066 N/A 0.0524 52.147 0.134
MRK-nu-1 GDSC1000 2.841 N/A 6.6 94.317 0
HCC1569 GDSC1000 22.313 N/A 0.0423 53.080 0.137
MCF7 GDSC1000 2.526 N/A 0.146 88.630 0.00132
HCC1187 GDSC1000 11.588 N/A 1e-06 88.412 0.0176
MDA-MB-175-VII GDSC1000 31.587 0.246 0.198 10.891 0.284
CAL-120 GDSC1000 8.375 2.29e+03 2.29e+03 0.000 0
HCC1806 GDSC1000 9.655 N/A 0.099 76.801 0.0536
MDA-MB-436 GDSC1000 10.312 2.52e+11 1.96e+03 46.227 0
EVSA-T GDSC1000 2.662 N/A 0.152 87.593 0.00272
ZR-75-30 GDSC1000 31.361 0.243 0.0287 40.480 0.256
HCC38 GDSC1000 2.861 N/A 0.0696 93.614 0
HCC38 GDSC1000 4.121 N/A 0.521 91.758 0
AU565 GDSC1000 45.025 0.0277 0.0167 25.960 0.396
HCC1143 GDSC1000 18.469 N/A 1.51e-05 63.062 0
MDA-MB-436 GDSC1000 4.918 N/A 0.0114 92.783 0
HCC1954 GDSC1000 23.901 3.11 0.0659 47.386 0.182
BT-483 GDSC1000 0.000 N/A 0.0391 100.000 0
MRK-nu-1 GDSC1000 0.593 N/A 0.000646 99.319 0
HCC1428 GDSC1000 1.465 N/A 0.0352 96.940 0
HCC202 GDSC1000 18.001 0.239 0.0856 43.851 0.139
HCC202 GDSC1000 22.899 0.856 0.225 33.806 0.183
MDA-MB-468 GDSC1000 20.469 N/A 0.0304 59.477 0.158
CAL-120 GDSC1000 9.482 N/A 1e+06 81.036 0
HCC2157 GDSC1000 30.063 0.13 0.0546 27.468 0.234
BT-483 GDSC1000 3.061 N/A 0.496 93.878 0
ZR-75-30 GDSC1000 31.729 N/A 0.0127 51.800 0.252
HDQ-P1 GDSC1000 22.966 N/A 0.0323 53.550 0.161
MDA-MB-175-VII GDSC1000 45.096 0.0274 0.0208 21.304 0.408
HCC1500 GDSC1000 0.187 22.8 16.3 36.836 0
HCC1569 GDSC1000 20.461 746 746 0.000 0
CAL-85-1 GDSC1000 7.266 N/A 405 85.468 0
JIMT-1 GDSC1000 8.865 N/A 1.37 53.989 0.0532
BT-474 GDSC1000 28.608 0.578 0.0633 37.680 0.226
MFM-223 GDSC1000 3.859 N/A 0.142 92.282 0
BT-549 GDSC1000 6.309 N/A 0.0652 86.099 0.0176
BT-549 GDSC1000 0.793 N/A 0.0895 97.636 0
MDA-MB-330 GDSC1000 30.084 N/A 0.0099 57.089 0.231
MCF7 GDSC1000 1.480 N/A 0.102 97.039 0
AU565 GDSC1000 30.284 0.149 0.0834 29.837 0.27
MDA-MB-361 GDSC1000 14.016 N/A 0.35 54.434 0.0946
MDA-MB-361 GDSC1000 11.879 N/A 0.0313 76.234 0.0683
DU-4475 GDSC1000 0.844 N/A 0.175 95.547 0
MDA-MB-157 GDSC1000 6.761 1.89e+18 1e+06 48.023 0
HCC2157 GDSC1000 5.456 13.7 13.7 0.000 0
EFM-192A GDSC1000 22.818 1.2 0.143 40.959 0.178
EFM-192A GDSC1000 48.538 0.0249 0.0156 21.053 0.43
MDA-MB-330 GDSC1000 17.186 N/A 0.0736 61.203 0.124
HCC1500 GDSC1000 3.621 N/A 0.0369 92.300 0
DU-4475 GDSC1000 1.830 N/A 0.0936 96.340 0
HCC1187 GDSC1000 2.270 N/A 0.0999 95.460 0
OCUB-M GDSC1000 4.658 N/A 0.155 78.015 0.0207
HCC1428 GDSC1000 0.000 N/A 0.0391 100.000 0
CAL-51 GDSC1000 4.830 N/A 0.0655 89.830 0.0715
MDA-MB-453 GDSC1000 4.749 N/A 1e+06 53.797 0
EVSA-T GDSC1000 0.020 N/A 2.5 99.862 0
COLO-824 GDSC1000 5.779 N/A 0.0025 93.859 0
CAL-85-1 GDSC1000 19.853 N/A 0.0543 57.812 0.145
MDA-MB-415 GDSC1000 9.861 N/A 0.0136 80.278 0
HCC1395 GDSC1000 1.639 N/A 0.782 92.870 0
MDA-MB-415 GDSC1000 1.090 N/A 0.145 95.133 0
HCC1954 GDSC1000 5.037 N/A 0.027 90.434 0
HCC1395 GDSC1000 0.000 N/A 0.00195 100.000 0
MDA-MB-468 GDSC1000 16.572 N/A 0.0986 60.232 0.12
COLO-824 GDSC1000 4.229 2.11e+03 2.11e+03 0.000 0
T47D GDSC1000 14.434 N/A 0.105 66.984 0.0634
HCC1143 GDSC1000 17.268 N/A 0.0158 72.153 0.102
JIMT-1 GDSC1000 7.156 N/A 0.167 65.698 0.0357
MDA-MB-453 GDSC1000 7.987 36.6 2.44 46.312 0.0477
OCUB-M GDSC1000 22.443 0.733 0.481 18.747 0.192
CAL-51 GDSC1000 1.850 23 23 0.000 0
BT-474 GRAY 58.002 0.024 0.0185 8.278 0.539
BT-474 GRAY 51.975 0.0492 0.0349 11.174 0.478
CAMA-1 GRAY 21.960 3.67 3.61 3.037 0.212
HCC1143 GRAY 31.282 1.38 1.38 0.000 0.268
HCC1395 GRAY 24.860 2.75 2.73 0.460 0.225
HCC2185 GRAY 19.999 5.21 5.21 0.000 0.179
MDA-MB-134-VI GRAY 18.441 6.38 6.38 0.000 0.164
MDA-MB-175-VII GRAY 53.219 0.0536 0.0481 5.271 0.502
MDA-MB-231 GRAY 30.480 1.75 1.75 0.000 0.253
MX-1 GRAY 26.298 2.14 2.08 2.388 0.247
SUM225CWN GRAY 48.739 0.113 0.0891 4.887 0.433
BT-20 GRAY 23.009 3.63 3.63 0.000 0.203
BT-483 GRAY 18.391 7.24 7.24 0.000 0.154
HCC1428 GRAY 20.435 4.93 4.93 0.000 0.183
HCC1937 GRAY 26.382 2.64 2.64 0.000 0.223
HCC1954 GRAY 42.973 0.262 0.25 1.452 0.387
HCC38 GRAY 25.226 2.61 2.61 0.000 0.232
MCF10A GRAY 52.953 0.04 0.0341 10.045 0.504
SK-BR-3 GRAY 56.322 0.0217 0.018 11.783 0.536
SUM 149PT GRAY 46.428 0.178 0.178 0.000 0.411
SUM 159PT GRAY 25.177 2.63 2.63 0.000 0.233
SUM 229PE GRAY 31.480 1.39 1.39 0.000 0.267
SUM 52PE GRAY 20.195 4.78 4.65 2.472 0.187
UACC-812 GRAY 47.088 0.162 0.162 0.000 0.418
ZR75B GRAY 22.377 3.75 3.75 0.000 0.21
184A1 GRAY 51.722 0.0431 0.0279 14.144 0.475
184B5 GRAY 44.577 0.231 0.231 0.000 0.393
600MPE GRAY 21.668 4.1 4.1 0.000 0.204
BT-474 GRAY 60.187 0.0194 0.0156 6.410 0.56
BT-549 GRAY 28.462 1.74 1.74 0.000 0.26
HCC1395 GRAY 22.442 3.9 3.9 0.000 0.198
HCC1419 GRAY 50.012 0.0667 0.0435 11.854 0.453
HCC1569 GRAY 27.545 3.23 3.23 0.000 0.218
HCC1806 GRAY 31.542 1.28 1.28 0.000 0.274
HCC70 GRAY 31.598 1.25 1.25 0.000 0.276
Hs-578-T GRAY 23.447 2.66 2.48 8.318 0.222
LY2 GRAY 24.381 2.66 2.62 3.073 0.235
MB 157 GRAY 60.079 0.0177 0.0131 8.223 0.558
MCF10F GRAY 41.979 0.322 0.322 0.000 0.371
MCF12A GRAY 43.963 0.192 0.156 6.736 0.398
MDA-MB-157 GRAY 22.948 3.25 3.2 2.754 0.221
MDA-MB-231 GRAY 19.713 4.95 4.87 3.032 0.189
MDA-MB-361 GRAY 40.368 0.4 0.4 0.000 0.356
MDA-MB-415 GRAY 25.024 2.68 2.68 0.000 0.231
MDA-MB-453 GRAY 39.146 0.468 0.468 0.000 0.345
SUM 1315M02 GRAY 25.964 3.6 3.6 0.000 0.207
SUM185PE GRAY 18.462 5.24 5.01 8.174 0.176
T47D_KBluc GRAY 20.133 4.75 4.69 2.333 0.194
ZR-75-1 GRAY 21.338 4.78 4.78 0.000 0.182
BT-474 FIMM 52.955 0.0449 0.0209 18.003 0.477
BT-549 FIMM 11.662 3.64 3.64 0.000 0.0977
CAL-120 FIMM 39.173 0.676 0.676 0.000 0.324
HCC1143 FIMM 32.807 10.4 10.4 0.000 0
HCC1599 FIMM 15.046 1.16e+06 1e+06 0.778 0
HCC1937 FIMM 19.899 1.9 1.9 0.000 0.162
Hs-578-T FIMM 10.065 4.26 4.26 0.000 0.0828
MCF7 FIMM 24.010 2.69 2.69 0.000 0.172
MDA-MB-231 FIMM 18.216 1.99 1.99 0.000 0.156
MDA-MB-436 FIMM 8.108 4.6 4.22 14.375 0.0701
MDA-MB-468 FIMM 32.527 0.693 0.693 0.000 0.264
MFM-223 FIMM 14.093 3.73 3.73 0.000 0.106
SK-BR-3 FIMM 66.176 0.0103 0.00753 14.012 0.624
T47D FIMM 16.604 9.72 9.72 0.000 0.101
ZR-75-1 FIMM 30.717 0.00242 0.00242 0.000 0.23
CAL-148 FIMM 25.424 5.7 5.7 0.000 0.174
CAL-51 FIMM 2.937 10.1 9.7 4.960 0.0173
CAL-85-1 FIMM 41.703 0.302 0.302 0.000 0.352
DU-4475 FIMM 12.093 166 166 0.000 0
HDQ-P1 FIMM 31.588 0.667 0.667 0.000 0.262
MDA-MB-453 FIMM 47.460 0.0891 0.055 15.398 0.422
KPL-1 CTRPv2 18.008 10.1 10.1 0.000 0.171
HDQ-P1 CTRPv2 37.637 1.57 1.57 0.000 0.32
JIMT-1 CTRPv2 20.964 6.5 6.24 7.504 0.199
HARA CTRPv2 35.560 2.22 2.22 0.000 0.294
CAMA-1 CTRPv2 11.595 65.4 65.4 0.000 0.0688
MCF7 CTRPv2 28.758 3.98 3.98 0.000 0.24
HCC1806 CTRPv2 34.269 2.11 2.11 0.000 0.294
HCC1954 CTRPv2 57.134 0.146 0.137 1.487 0.524
HMC-1-8 CTRPv2 23.020 5.93 5.87 1.085 0.214
HCC1937 CTRPv2 22.580 8.68 8.68 0.000 0.179
CAL-148 CTRPv2 29.601 2.92 2.84 2.168 0.275
CAL-51 CTRPv2 24.489 4.35 4.17 7.748 0.234
HCC1395 CTRPv2 16.265 12.9 12.9 0.000 0.14
MDA-MB-231 CTRPv2 28.139 3.89 3.89 0.000 0.242
HCC1143 CTRPv2 40.059 1.22 1.22 0.000 0.341
ZR-75-1 CTRPv2 27.641 1.6 1.32 26.455 0.258
HCC1428 CTRPv2 21.148 8.2 8.2 0.000 0.178
HCC38 CTRPv2 24.058 7.1 7.1 0.000 0.194
BT-549 CTRPv2 17.129 11 8.96 12.640 0.145
HCC202 CTRPv2 44.409 0.792 0.792 0.000 0.382
HCC1500 CTRPv2 28.453 2.92 2.82 6.072 0.274
Hs-578-T CTRPv2 30.804 2.57 2.52 1.827 0.29
MDA-MB-468 CTRPv2 46.093 0.572 0.572 0.000 0.407
CAL-85-1 CTRPv2 53.258 0.205 0.205 0.000 0.481
BT-20 CTRPv2 20.264 6.28 5.81 13.220 0.191
UACC-812 CTRPv2 55.417 0.0436 0.0177 28.834 0.505
HCC1419 CTRPv2 26.246 N/A 0.0948 58.183 0.199
ZR-75-30 CTRPv2 72.677 0.00873 0.00533 14.254 0.696
MDA-MB-157 CTRPv2 40.381 1.11 1.11 0.000 0.349
MDA-MB-361 CTRPv2 47.598 0.596 0.596 0.000 0.418
T47D CTRPv2 22.737 6.73 6.73 0.000 0.195
BT-474 CTRPv2 53.556 0.225 0.225 0.000 0.484
HCC2218 CTRPv2 74.085 0.0102 0.0078 13.196 0.712
SK-BR-3 CTRPv2 67.884 0.00662 0.00275 24.180 0.643
MDA-MB-453 CTRPv2 26.339 4.28 4.28 0.000 0.244
AU565 CTRPv2 61.721 0.0669 0.0648 0.590 0.575
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