Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MEL-HO GDSC1000 29.416 0.667 0.667 0.000 0.221
A375 GDSC1000 34.370 0.307 0.243 11.953 0.289
CP50-MEL-B GDSC1000 25.147 0.764 0.439 19.754 0.187
Hs 939.T GDSC1000 23.229 0.774 0.494 18.760 0.174
IGR-37 GDSC1000 43.142 0.181 0.156 7.105 0.375
A101D GDSC1000 27.842 0.402 0.265 24.453 0.232
SK-MEL-31 GDSC1000 7.627 N/A 0.599 66.922 0.0365
GAK GDSC1000 25.025 1.88 1.88 0.000 0.168
A388 GDSC1000 22.337 0.764 0.19 47.452 0.177
COLO-783 GDSC1000 5.203 N/A 0.933 62.751 0.0317
WM-115 GDSC1000 27.196 0.414 0.164 39.883 0.221
WM793B GDSC1000 17.175 1.44 1.44 0.000 0.112
COLO-679 GDSC1000 10.536 N/A 0.552 54.926 0.0748
COLO-800 GDSC1000 24.335 0.707 0.707 0.000 0.185
MZ2-MEL GDSC1000 42.319 0.171 0.141 11.626 0.374
WM239A GDSC1000 12.643 2.15 2.15 0.000 0
MCC26 GDSC1000 11.110 2.25 1.5 18.646 0.0651
MEL-JUSO GDSC1000 25.418 0.746 0.234 36.096 0.192
WM1552C GDSC1000 41.137 3.68 3.68 0.000 0
LB2518-MEL GDSC1000 17.083 2.9 2.9 0.000 0
IST-MEL1 GDSC1000 13.388 1.03 0.714 29.915 0.105
IGR-1 GDSC1000 8.828 2.55 2.55 0.000 0
SH-4 GDSC1000 31.776 1.19 1.19 0.000 0.242
451Lu GDSC1000 27.673 0.387 0.26 25.276 0.234
SK-MEL-2 GDSC1000 21.786 0.841 0.633 12.936 0.162
SK-MEL-3 GDSC1000 14.483 1.86 0.727 34.076 0.095
SK-MEL-5 GDSC1000 28.589 0.431 0.23 27.865 0.231
WM35 GDSC1000 28.983 0.513 0.513 0.000 0.229
CHL-1 GDSC1000 33.588 0.311 0.285 5.903 0.292
IPC-298 GDSC1000 20.719 1.03 1.03 0.000 0.146
A253 GDSC1000 10.592 1.81 0.883 36.632 0.0712
RPMI-7951 GDSC1000 22.613 0.762 0.716 3.149 0.171
C32 GDSC1000 20.909 1.39 0.401 34.971 0.145
DJM-1 GDSC1000 25.066 1.82 1.82 0.000 0.169
HT-144 GDSC1000 30.340 1.35 0.0788 47.052 0.231
A431 GDSC1000 32.626 0.841 0.841 0.000 0.251
MZ7-mel GDSC1000 17.586 N/A 0.158 61.614 0.127
RVH-421 GDSC1000 27.148 0.648 0.648 0.000 0.206
LB373-MEL-D GDSC1000 7.952 N/A 0.766 56.846 0.0466
SK-MEL-1 GDSC1000 14.927 N/A 0.39 51.107 0.0992
CP66-MEL GDSC1000 18.250 2.44 0.335 45.696 0.126
G-361 GDSC1000 34.469 0.45 0.16 26.030 0.273
RPMI-7951 CTRPv2 45.798 0.134 0.048 33.817 0.406
A375 CTRPv2 36.077 0.144 0.0866 43.438 0.323
MEL-HO CTRPv2 56.099 0.0907 0.0592 16.279 0.517
SK-MEL-1 CTRPv2 30.449 N/A 0.0847 52.398 0.249
Hs 944.T CTRPv2 37.190 1.16 0.0476 45.736 0.306
MEL-JUSO CTRPv2 42.274 0.25 0.0777 34.560 0.37
SK-MEL-31 CTRPv2 24.204 N/A 0.0539 62.781 0.16
SK-MEL-5 CTRPv2 41.763 0.288 0.141 29.302 0.374
IPC-298 CTRPv2 41.129 0.312 0.0875 35.159 0.357
SK-MEL-30 CTRPv2 29.674 1 0.191 47.174 0.252
A375 CTRPv2 28.997 N/A 0.0123 64.558 0.216
WM1799 CTRPv2 38.290 N/A 0.0137 50.695 0.314
WM-793 CTRPv2 40.087 0.571 0.113 33.820 0.34
G-361 CTRPv2 47.634 0.12 0.0301 34.658 0.42
Hs 852.T CTRPv2 50.610 0.0275 0.00621 42.103 0.451
Hs 936.T CTRPv2 28.769 N/A 0.0916 54.289 0.223
COLO-800 CTRPv2 32.089 399 0.0717 49.460 0.247
K029AX CTRPv2 40.421 1.16 0.0451 39.196 0.338
COLO-829 CTRPv2 39.924 0.744 0.0246 43.858 0.332
IGR-1 CTRPv2 51.504 0.169 0.0681 11.104 0.461
SH-4 CTRPv2 48.500 0.035 0.0133 39.530 0.432
A253 CTRPv2 38.794 0.618 0.0374 45.317 0.324
C32 CTRPv2 36.202 N/A 0.00866 55.312 0.291
HT-144 CTRPv2 38.533 1.19 0.066 40.296 0.318
Hs 294T CTRPv2 53.758 0.069 0.0193 28.740 0.486
SK-MEL-2 CTRPv2 6.105 56.8 56.8 0.000 0.0384
A101D CTRPv2 34.309 N/A 0.0373 52.066 0.28
A2058 CTRPv2 38.365 0.547 0.129 35.723 0.328
COLO-792 CTRPv2 50.745 0.271 0.185 8.697 0.453
HMCB CTRPv2 43.026 0.176 0.0307 41.170 0.371
IGR-39 CTRPv2 45.316 0.224 0.0256 37.967 0.392
Mewo CTRPv2 46.683 0.127 0.0158 40.079 0.408
WM-115 CTRPv2 43.175 0.769 0.032 36.283 0.369
WM-266-4 CTRPv2 47.985 0.174 0.0172 35.808 0.422
Hs 895.T CTRPv2 49.896 0.0634 0.00373 42.491 0.443
SK-MEL-24 CTRPv2 30.222 6.67 0.277 42.298 0.235
RVH-421 CTRPv2 35.621 1.21 0.0714 45.282 0.293
Hs 839.T CTRPv2 27.386 N/A 0.0168 64.709 0.201
WM-88 CTRPv2 60.973 0.0168 0.00863 26.959 0.566
WM-983B CTRPv2 32.910 1.46 0.11 43.626 0.266
CJM CTRPv2 31.182 1.37 0.289 40.256 0.261
SK-MEL-3 CTRPv2 42.352 0.478 0.0352 39.442 0.36
IGR-37 CTRPv2 31.788 7.57 0.201 42.132 0.247
Hs 934.T CTRPv2 22.498 N/A 0.0126 72.131 0.148
Hs 688(A).T CTRPv2 20.760 N/A 0.0701 68.358 0.138
Hs 940.T CTRPv2 41.848 0.196 0.0161 47.163 0.357
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