Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
MEL-HO GDSC1000 24.863 0.579 0.188 41.916 0.196
A375 GDSC1000 43.874 0.176 0.174 0.909 0.395
A431 GDSC1000 18.533 0.699 0.4 36.475 0.15
G-MEL GDSC1000 51.165 0.106 0.1 5.168 0.475
COLO-800 GDSC1000 22.010 0.627 0.559 8.816 0.182
SK-MEL-31 GDSC1000 33.224 0.366 0.16 27.976 0.267
WM35 GDSC1000 31.839 0.46 0.46 0.000 0.252
WM278 GDSC1000 39.587 0.189 0.15 15.372 0.35
MCC26 GDSC1000 28.234 0.61 0.61 0.000 0.215
SK-MEL-3 GDSC1000 9.104 N/A 0.595 58.451 0.0654
A101D GDSC1000 28.538 0.379 0.213 29.839 0.236
WM793B GDSC1000 29.887 0.263 0.217 25.314 0.272
Mewo GDSC1000 33.776 0.24 0.185 21.350 0.3
451Lu GDSC1000 34.510 0.228 0.184 19.863 0.31
MMAC-SF GDSC1000 10.695 N/A 0.00308 78.611 0
COLO-679 GDSC1000 45.234 0.119 0.11 13.414 0.429
CP66-MEL GDSC1000 18.515 0.683 0.321 43.948 0.15
VMRC-MELG GDSC1000 5.750 12.7 12.7 0.000 0
G-361 GDSC1000 51.872 0.0896 0.0435 16.297 0.465
SK-MEL-30 GDSC1000 35.955 0.278 0.224 10.864 0.304
MEL-JUSO GDSC1000 45.415 0.15 0.123 9.650 0.399
IST-MEL1 GDSC1000 39.699 0.179 0.109 24.270 0.342
COLO-783 GDSC1000 34.440 0.187 0.131 29.880 0.306
HMV-II GDSC1000 22.134 631 631 0.000 0
RPMI-7951 GDSC1000 35.337 0.237 0.217 11.834 0.327
WM-115 GDSC1000 6.738 2.87 1.48 34.114 0.0366
DJM-1 GDSC1000 21.658 0.692 0.373 30.454 0.17
LB373-MEL-D GDSC1000 0.206 4.3 4.3 0.000 0
A2058 GDSC1000 30.185 0.415 0.415 0.000 0.253
SK-MEL-2 GDSC1000 55.523 0.0602 0.0466 17.483 0.51
IPC-298 GDSC1000 47.529 0.12 0.108 9.746 0.438
A388 GDSC1000 14.106 1.08 0.566 39.020 0.108
LB2518-MEL GDSC1000 7.933 N/A 0.77 54.639 0.0539
WM1158 GDSC1000 41.235 0.212 0.212 0.000 0.361
SK-MEL-24 GDSC1000 13.390 5.41 5.41 0.000 0
CP50-MEL-B GDSC1000 0.000 N/A 0.00781 100.000 0
A253 GDSC1000 25.787 0.628 0.628 0.000 0.2
RVH-421 GDSC1000 16.585 0.799 0.4 43.000 0.133
SK-MEL-5 GDSC1000 29.893 0.498 0.498 0.000 0.236
SH-4 GDSC1000 9.272 1.22 1.01 26.421 0.0747
Hs 939.T GDSC1000 30.746 0.472 0.355 11.047 0.243
C32 GDSC1000 45.624 0.0891 0.0715 24.051 0.42
IGR-37 GDSC1000 62.734 0.0552 0.0527 3.520 0.589
MCC13 GDSC1000 7.402 6.35 6.35 0.000 0
CHL-1 GDSC1000 24.463 0.465 0.36 21.380 0.21
WM1552C GDSC1000 18.374 1.26 0.447 36.514 0.131
IGR-1 GDSC1000 5.140 2.84 1.18 48.492 0.0339
SK-MEL-1 GDSC1000 0.211 4.99 3.88 31.806 0
GAK GDSC1000 15.765 0.824 0.495 37.738 0.127
MZ2-MEL GDSC1000 11.641 2.27 2.27 0.000 0
RPMI-7951 CTRPv2 61.572 0.0873 0.0795 4.301 0.58
A375 CTRPv2 49.711 0.321 0.306 3.780 0.473
MEL-HO CTRPv2 33.068 2.36 2.36 0.000 0.285
SK-MEL-1 CTRPv2 25.831 3.18 2.17 21.404 0.229
Hs 944.T CTRPv2 59.027 0.0468 0.0256 20.677 0.545
MEL-JUSO CTRPv2 46.654 0.224 0.203 16.073 0.448
SK-MEL-31 CTRPv2 25.581 11.2 11.2 0.000 0.188
SK-MEL-5 CTRPv2 25.293 5.55 5.55 0.000 0.212
IPC-298 CTRPv2 41.761 0.223 0.186 26.023 0.393
SK-MEL-30 CTRPv2 30.024 4 4 0.000 0.244
A375 CTRPv2 39.236 1.43 1.43 0.000 0.33
WM1799 CTRPv2 41.234 1 1 0.000 0.358
WM-793 CTRPv2 41.383 0.915 0.915 0.000 0.373
G-361 CTRPv2 41.775 0.663 0.419 14.216 0.367
Hs 852.T CTRPv2 52.864 0.202 0.157 8.333 0.482
Hs 936.T CTRPv2 42.545 0.366 0.0643 35.116 0.364
COLO-800 CTRPv2 39.688 0.287 0.175 30.401 0.361
K029AX CTRPv2 25.543 5.1 5.1 0.000 0.219
COLO-829 CTRPv2 41.023 0.785 0.525 12.080 0.359
IGR-1 CTRPv2 39.231 1.17 1.15 0.473 0.347
SH-4 CTRPv2 39.076 1.39 1.39 0.000 0.331
A253 CTRPv2 34.181 1.82 1.66 4.170 0.305
C32 CTRPv2 51.912 0.239 0.197 6.666 0.474
HT-144 CTRPv2 31.337 2.65 2.65 0.000 0.278
Hs 294T CTRPv2 43.696 0.706 0.706 0.000 0.402
SK-MEL-2 CTRPv2 26.647 0.71 0.338 47.426 0.233
A101D CTRPv2 36.742 1.67 1.67 0.000 0.314
A2058 CTRPv2 44.914 0.425 0.406 8.206 0.436
COLO-792 CTRPv2 18.861 12.9 12.9 0.000 0.147
HMCB CTRPv2 45.488 0.418 0.402 7.212 0.442
IGR-39 CTRPv2 45.952 0.557 0.557 0.000 0.424
Mewo CTRPv2 39.873 0.426 0.375 19.755 0.38
WM-115 CTRPv2 31.705 2.69 2.69 0.000 0.274
WM-266-4 CTRPv2 34.257 1.92 1.92 0.000 0.309
Hs 895.T CTRPv2 42.756 0.854 0.854 0.000 0.372
SK-MEL-24 CTRPv2 29.826 3.04 3.04 0.000 0.269
RVH-421 CTRPv2 33.857 2.27 2.27 0.000 0.288
Hs 839.T CTRPv2 39.201 1.51 1.51 0.000 0.328
WM-88 CTRPv2 41.272 0.621 0.459 13.592 0.374
WM-983B CTRPv2 45.192 0.286 0.146 22.839 0.404
CJM CTRPv2 39.982 1.03 1.03 0.000 0.376
SK-MEL-3 CTRPv2 24.681 5.8 5.8 0.000 0.208
IGR-37 CTRPv2 40.273 0.274 0.228 26.075 0.379
Hs 934.T CTRPv2 37.864 1.53 1.53 0.000 0.322
Hs 688(A).T CTRPv2 29.121 3.75 3.75 0.000 0.245
Hs 940.T CTRPv2 42.766 0.793 0.793 0.000 0.385
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