Summary Statistics

Cell Line DatasetAAC (%)IC50 (µM)EC50 (µM)Einf (%)DSS1 (arb.)
AU565 CCLE 56.417 0.0224 0.0143 27.765 0.52
BT-20 CCLE 20.861 177 177 0.000 0
BT-474 CCLE 63.141 0.0347 0.0307 8.101 0.597
BT-549 CCLE 62.160 0.0215 0.0127 19.635 0.58
CAL-85-1 CCLE 45.217 0.201 0.14 9.763 0.392
CAMA-1 CCLE 47.039 0.12 0.0181 32.708 0.412
EFM-19 CCLE 45.772 0.0576 0.0401 30.249 0.42
HARA CCLE 38.220 0.2 0.163 20.718 0.356
HCC1187 CCLE 13.610 1.9 1.22 41.704 0.116
HCC1395 CCLE 32.465 N/A 0.00981 60.721 0.255
HCC1569 CCLE 39.015 0.198 0.138 22.383 0.353
HCC1806 CCLE 53.108 0.0694 0.0653 10.861 0.513
HCC1954 CCLE 59.033 0.0402 0.0299 13.913 0.547
HCC70 CCLE 45.654 0.122 0.0635 23.232 0.403
HDQ-P1 CCLE 40.080 0.114 0.0888 28.128 0.371
HMC-1-8 CCLE 49.998 0.0922 0.0765 13.188 0.466
Hs-578-T CCLE 49.802 0.0553 0.0444 22.598 0.467
Hs 739.T CCLE 26.610 0.568 0.375 29.843 0.235
MB 157 CCLE 34.878 0.132 0.094 36.662 0.317
MCF7 CCLE 52.148 0.115 0.115 0.000 0.468
MDA-MB-157 CCLE 10.913 N/A 0.0274 84.486 0.0378
MDA-MB-175-VII CCLE 46.279 0.0295 0.021 37.127 0.423
MDA-MB-415 CCLE 65.574 0.0177 0.0157 15.104 0.629
MDA-MB-436 CCLE 29.265 N/A 0.0463 54.096 0.234
MDA-MB-453 CCLE 73.969 0.0168 0.0164 3.518 0.725
MDA-MB-468 CCLE 26.328 0.539 0.228 40.267 0.224
SK-BR-3 CCLE 47.154 0.0237 0.00737 45.114 0.414
T47D CCLE 16.683 1.78 1.07 33.235 0.14
UACC-812 CCLE 48.665 0.127 0.0347 21.678 0.43
ZR-75-1 CCLE 60.516 0.0369 0.0287 12.473 0.564
ZR-75-30 CCLE 37.155 0.0955 0.0455 41.988 0.327
HDQ-P1 GDSC1000 17.630 0.453 0.274 28.140 0.135
MDA-MB-231 GDSC1000 1.889 N/A 0.295 91.423 0
UACC-893 GDSC1000 30.567 0.924 0.924 0.000 0.229
CAL-51 GDSC1000 61.562 0.0259 0.0248 7.657 0.594
HARA GDSC1000 41.990 0.0695 0.0411 26.683 0.366
HCC2218 GDSC1000 34.704 N/A 0.019 51.448 0.294
CAL-120 GDSC1000 16.998 0.518 0.384 16.703 0.125
HCC1954 GDSC1000 16.769 N/A 0.0775 63.642 0.124
MRK-nu-1 GDSC1000 0.396 N/A 0.279 98.284 0
HCC1569 GDSC1000 21.627 N/A 0.0385 61.621 0.132
MDA-MB-453 GDSC1000 34.068 1.04 0.0233 45.153 0.267
MCF7 GDSC1000 51.590 0.0148 0.0106 37.059 0.469
EVSA-T GDSC1000 51.479 0.0298 0.0238 23.603 0.476
DU-4475 GDSC1000 28.121 0.214 0.214 0.000 0.251
HCC38 GDSC1000 25.625 0.241 0.123 32.777 0.207
MDA-MB-468 GDSC1000 0.442 1.77 1.77 0.000 0
BT-483 GDSC1000 19.679 N/A 0.0363 67.048 0.134
MDA-MB-361 GDSC1000 60.091 0.022 0.0174 17.014 0.558
HCC1806 GDSC1000 35.459 0.0846 0.057 31.358 0.314
HCC1937 GDSC1000 34.113 0.0984 0.0391 41.561 0.287
HCC1187 GDSC1000 2.099 N/A 0.0778 95.443 0
HCC1500 GDSC1000 9.011 4.74 4.74 0.000 0
CAL-85-1 GDSC1000 5.894 N/A 1e+06 88.212 0
JIMT-1 GDSC1000 50.410 0.0422 0.0346 16.757 0.464
MDA-MB-157 GDSC1000 41.077 0.0328 0.0153 45.411 0.357
HCC2157 GDSC1000 42.673 0.0783 0.0574 17.074 0.375
AU565 GDSC1000 42.744 0.0253 0.00953 48.989 0.37
EFM-192A GDSC1000 47.571 0.0368 0.00885 40.888 0.417
T47D GDSC1000 7.472 N/A 0.0089 91.209 0
MDA-MB-330 GDSC1000 53.617 0.016 0.00451 39.378 0.485
HCC1419 GDSC1000 34.150 0.0751 0.0371 42.491 0.294
MFM-223 GDSC1000 29.239 0.212 0.0409 49.275 0.241
HCC1428 GDSC1000 24.485 N/A 0.0156 67.318 0.175
BT-549 GDSC1000 38.683 0.0899 0.0513 27.587 0.332
COLO-824 GDSC1000 39.720 0.18 0.121 8.371 0.33
Hs-578-T GDSC1000 44.803 0.0447 0.0254 32.021 0.395
HCC1395 GDSC1000 14.682 N/A 0.0463 73.367 0.0762
MDA-MB-436 GDSC1000 35.724 0.0839 0.0571 30.800 0.317
OCUB-M GDSC1000 1.724 1.21 1.21 0.000 0
BT-20 GDSC1000 32.918 N/A 0.0118 58.754 0.263
MDA-MB-415 GDSC1000 31.289 N/A 0.0245 52.172 0.241
HCC202 GDSC1000 12.352 N/A 0.0751 73.540 0.0766
BT-474 GDSC1000 55.144 0.0146 0.00676 36.264 0.502
ZR-75-30 GDSC1000 23.130 N/A 0.0599 54.439 0.187
HCC1143 GDSC1000 35.272 0.173 0.0781 24.449 0.284
184A1 GRAY 42.023 0.0291 0.0203 36.360 0.387
600MPE GRAY 35.381 1.5 1.5 0.000 0.293
BT-474 GRAY 46.163 0.0469 0.0309 26.464 0.429
BT-474 GRAY 32.396 N/A 0.0143 52.884 0.278
BT-483 GRAY 22.138 9.56 9.56 0.000 0.172
HCC1395 GRAY 30.226 2.93 2.93 0.000 0.247
HCC1419 GRAY 38.287 0.211 0.135 25.393 0.352
HCC1419 GRAY 47.503 0.076 0.0596 17.634 0.449
HCC1569 GRAY 38.472 0.248 0.154 23.490 0.352
HCC1954 GRAY 48.172 0.0536 0.0385 21.123 0.452
HCC202 GRAY 37.619 1.21 1.21 0.000 0.311
HCC202 GRAY 35.757 1.45 1.45 0.000 0.296
HCC2185 GRAY 32.976 0.495 0.202 31.583 0.291
HCC2185 GRAY 28.203 0.901 0.406 34.063 0.249
HCC38 GRAY 37.044 0.225 0.141 27.304 0.34
HCC70 GRAY 40.133 0.324 0.23 14.926 0.368
Hs-578-T GRAY 41.780 0.186 0.152 17.099 0.396
LY2 GRAY 44.534 0.0784 0.0505 24.464 0.413
LY2 GRAY 41.045 0.175 0.14 19.594 0.388
MCF10A GRAY 55.066 0.0492 0.0453 7.909 0.532
MCF7 GRAY 26.026 8.05 8.05 0.000 0.197
MDA-MB-134-VI GRAY 36.526 0.491 0.207 23.942 0.319
MDA-MB-415 GRAY 41.249 0.129 0.108 22.250 0.391
MDA-MB-415 GRAY 48.574 0.0766 0.0479 18.120 0.447
MDA-MB-468 GRAY 28.721 1.7 1.57 10.966 0.274
MDA-MB-468 GRAY 27.595 1.99 1.88 10.650 0.266
SK-BR-3 GRAY 38.302 1.02 1.02 0.000 0.32
SUM102PT GRAY 23.517 N/A 0.0862 57.091 0.195
SUM 1315M02 GRAY 37.670 1.01 1.01 0.000 0.318
SUM 229PE GRAY 50.778 0.0333 0.0233 21.852 0.476
SUM 52PE GRAY 46.592 0.154 0.0976 13.299 0.42
UACC-812 GRAY 34.078 0.063 0.0241 47.320 0.3
ZR75B GRAY 34.055 0.65 0.134 33.675 0.288
ZR75B GRAY 40.964 0.11 0.0358 33.479 0.362
HCC1187 GRAY 23.841 2.71 2.19 19.675 0.221
HCC1395 GRAY 34.323 1.37 0.644 14.797 0.285
HCC1419 GRAY 35.696 0.471 0.266 22.507 0.321
HCC1806 GRAY 44.789 0.145 0.132 12.982 0.433
Hs-578-T GRAY 44.418 0.148 0.124 14.557 0.422
MCF10A GRAY 56.654 0.0469 0.045 5.343 0.553
MCF12A GRAY 51.511 0.0849 0.0803 6.936 0.501
MDA-MB-134-VI GRAY 48.636 0.0743 0.0654 14.593 0.467
MDA-MB-361 GRAY 44.095 0.111 0.0935 18.601 0.42
MDA-MB-436 GRAY 27.009 7.28 7.28 0.000 0.205
SUM 159PT GRAY 60.156 0.0315 0.0307 4.229 0.591
UACC-893 GRAY 49.270 0.0552 0.0483 16.915 0.473
184B5 GRAY 27.691 8.24 8.24 0.000 0.207
MCF12A GRAY 57.748 0.0472 0.0459 3.259 0.564
SUM 1315M02 GRAY 39.374 0.129 0.0623 31.304 0.356
SUM 229PE GRAY 43.814 0.137 0.0617 23.542 0.392
SUM44PE GRAY 50.030 0.112 0.0441 13.733 0.445
SUM 52PE GRAY 43.608 0.262 0.105 17.687 0.379
HCC1419 GRAY 46.105 0.254 0.191 5.559 0.404
HCC1954 GRAY 50.974 0.0591 0.0409 15.821 0.474
HCC1954 GRAY 49.041 0.0719 0.0636 14.205 0.472
HCC1954 GRAY 46.907 0.0716 0.0321 24.763 0.423
HCC1954 GRAY 30.600 3.79 3.79 0.000 0.241
HCC2185 GRAY 33.645 0.222 0.132 34.630 0.306
HCC2185 GRAY 37.815 0.658 0.333 15.325 0.324
HCC2185 GRAY 31.946 1.71 1.28 7.999 0.272
HCC38 GRAY 43.037 0.16 0.0751 22.885 0.385
HCC38 GRAY 40.950 0.15 0.0693 27.494 0.368
HCC70 GRAY 34.611 0.57 0.382 19.974 0.316
Hs-578-T GRAY 45.263 0.123 0.109 14.624 0.435
MCF10F GRAY 52.216 0.0531 0.0443 12.923 0.497
MDA-MB-134-VI GRAY 49.961 0.07 0.0621 12.878 0.481
MDA-MB-134-VI GRAY 42.170 0.111 0.0935 22.153 0.401
MDA-MB-175-VII GRAY 44.911 0.21 0.101 15.784 0.395
MDA-MB-231 GRAY 30.970 0.863 0.696 19.739 0.29
MDA-MB-361 GRAY 49.216 0.0589 0.0535 15.872 0.475
MDA-MB-361 GRAY 44.822 0.0783 0.0684 20.805 0.429
S1 GRAY 33.924 0.132 0.0872 38.002 0.309
SUM 149PT GRAY 53.562 0.0714 0.0689 5.282 0.523
SUM 149PT GRAY 58.407 0.0338 0.0256 8.328 0.542
SUM 159PT GRAY 55.336 0.0502 0.0481 6.749 0.541
184B5 GRAY 54.810 0.0345 0.0298 13.081 0.526
AU565 GRAY 37.493 1.12 1.12 0.000 0.313
AU565 GRAY 41.035 0.408 0.245 12.436 0.359
BT-483 GRAY 23.634 6.97 6.97 0.000 0.189
BT-549 GRAY 55.968 0.0255 0.0236 13.733 0.543
CAMA-1 GRAY 30.163 2.38 1.21 14.978 0.248
HCC1143 GRAY 35.594 0.209 0.142 30.089 0.329
HCC1143 GRAY 36.324 0.659 0.215 24.047 0.309
HCC1395 GRAY 28.414 4.14 4.14 0.000 0.227
HCC1395 GRAY 19.193 15 15 0.000 0.145
HCC1428 GRAY 27.431 6.13 6.13 0.000 0.211
HCC1428 GRAY 39.636 0.89 0.89 0.000 0.332
HCC1806 GRAY 45.041 0.0961 0.083 18.258 0.431
HCC2185 GRAY 34.709 0.948 0.629 12.454 0.304
HCC38 GRAY 20.846 N/A 0.0255 67.569 0.156
HCC38 GRAY 42.920 0.141 0.0951 20.576 0.398
HCC70 GRAY 29.085 0.944 0.569 27.549 0.263
MCF10A GRAY 58.021 0.0389 0.0373 5.363 0.567
MCF10F GRAY 59.113 0.0264 0.0252 8.143 0.578
MCF12A GRAY 56.232 0.0465 0.044 6.312 0.547
MCF7 GRAY 35.012 0.753 0.303 22.514 0.301
MDA-MB-175-VII GRAY 39.050 0.0997 0.0681 31.050 0.361
MDA-MB-231 GRAY 23.069 2.47 1.92 24.858 0.213
MDA-MB-231 GRAY 32.933 0.867 0.661 15.518 0.303
MDA-MB-361 GRAY 50.546 0.0495 0.0451 15.514 0.489
MDA-MB-436 GRAY 25.144 8.22 8.22 0.000 0.191
MDA-MB-436 GRAY 30.912 4.3 4.3 0.000 0.24
MDA-MB-453 GRAY 34.736 N/A 0.0119 50.528 0.303
MDA-MB-453 GRAY 45.415 0.0851 0.0757 18.624 0.436
MDA-MB-453 GRAY 49.012 0.0531 0.0399 19.373 0.462
MDA-MB-468 GRAY 26.570 2.05 1.89 13.781 0.254
SK-BR-3 GRAY 42.468 0.375 0.2 12.323 0.367
SK-BR-3 GRAY 31.721 46.6 0.0458 44.928 0.242
SUM 1315M02 GRAY 25.153 7.53 7.53 0.000 0.193
SUM 149PT GRAY 51.828 0.0834 0.0804 6.357 0.507
SUM 159PT GRAY 56.220 0.046 0.0433 6.535 0.546
SUM185PE GRAY 53.816 0.0385 0.0327 13.657 0.515
UACC-893 GRAY 53.440 0.0337 0.0218 18.300 0.497
UACC-893 GRAY 55.825 0.0328 0.0227 14.138 0.52
BT-549 GRAY 53.885 0.0442 0.0416 10.873 0.525
BT-549 GRAY 53.861 0.0411 0.0384 11.824 0.524
HBL-100 GRAY 29.405 1.95 1.81 5.585 0.275
HCC1187 GRAY 14.441 9.53 4.54 39.889 0.123
HCC1937 GRAY 42.155 0.128 0.112 20.070 0.403
HCC2185 GRAY 32.565 0.448 0.275 28.900 0.297
HCC3153 GRAY 36.717 0.224 0.153 27.088 0.34
HCC70 GRAY 27.425 2.38 1.41 17.813 0.237
MDA-MB-175-VII GRAY 43.005 0.109 0.0861 21.542 0.406
MDA-MB-453 GRAY 48.256 0.0545 0.0466 19.013 0.461
SUM185PE GRAY 44.945 0.0816 0.0676 20.723 0.427
ZR-75-1 GRAY 29.544 0.403 0.158 41.003 0.26
184A1 GRAY 19.505 9.85 9.85 0.000 0.161
600MPE GRAY 27.814 9.31 9.31 0.000 0.207
BT-549 GRAY 59.088 0.0246 0.0218 9.781 0.569
CAMA-1 GRAY 28.101 5.34 2.78 11.268 0.218
BT-483 GRAY 18.363 N/A 0.744 53.040 0.121
MB 157 GRAY 31.468 0.591 0.349 28.395 0.285
MCF10F GRAY 53.220 0.0508 0.0441 11.300 0.51
MDA-MB-361 GRAY 48.354 0.0774 0.0712 14.089 0.468
HBL-100 GRAY 34.820 0.973 0.903 4.774 0.326
HCC1395 GRAY 30.102 2.83 2.83 0.000 0.248
HCC1419 GRAY 36.858 0.708 0.385 15.238 0.319
HCC1419 GRAY 36.902 0.603 0.331 17.050 0.324
HCC1569 GRAY 39.792 0.202 0.145 21.616 0.371
HCC1937 GRAY 42.542 0.125 0.11 19.573 0.407
HCC1937 GRAY 40.223 0.166 0.129 22.170 0.378
HCC202 GRAY 34.928 1.51 1.38 1.941 0.29
HCC2185 GRAY 31.681 0.782 0.373 27.059 0.28
HCC70 GRAY 35.200 0.728 0.49 14.899 0.316
Hs-578-T GRAY 44.215 0.124 0.112 16.191 0.426
LY2 GRAY 39.498 0.114 0.0764 29.136 0.366
MCF10A GRAY 53.756 0.0524 0.0479 9.446 0.52
MCF10F GRAY 46.889 0.0833 0.0679 17.247 0.445
MCF7 GRAY 27.724 4.78 4.78 0.000 0.219
MDA-MB-157 GRAY 0.000 N/A 0.000256 100.000 0
MDA-MB-175-VII GRAY 42.774 0.144 0.073 23.708 0.386
MDA-MB-175-VII GRAY 41.821 0.126 0.0668 26.333 0.38
MDA-MB-361 GRAY 45.450 0.0654 0.0568 21.704 0.434
MDA-MB-436 GRAY 30.867 4.35 4.35 0.000 0.24
MDA-MB-468 GRAY 22.212 2.99 2.59 21.704 0.209
SK-BR-3 GRAY 39.435 1.01 1.01 0.000 0.328
SUM 1315M02 GRAY 24.642 N/A 0.0138 64.204 0.178
SUM 159PT GRAY 65.628 0.00939 0.00815 10.229 0.631
T47D GRAY 21.893 3.02 1.22 36.101 0.188
UACC-893 GRAY 46.023 0.0825 0.067 18.915 0.437
ZR-75-1 GRAY 30.349 0.209 0.137 40.737 0.275
BT-474 FIMM 40.859 0.0737 0.0612 26.148 0.384
BT-549 FIMM 49.529 0.0362 0.0219 25.382 0.452
CAL-120 FIMM 44.883 0.193 0.193 0.000 0.388
HCC1143 FIMM 53.553 0.0239 0.00884 27.983 0.484
HCC1599 FIMM 33.717 0.183 0.078 36.002 0.294
HCC1937 FIMM 40.274 0.0778 0.0644 26.469 0.378
Hs-578-T FIMM 44.219 0.104 0.0372 26.225 0.384
MCF7 FIMM 42.000 0.259 0.0587 22.532 0.356
MDA-MB-231 FIMM 19.691 0.99 0.803 28.099 0.179
MDA-MB-436 FIMM 51.159 0.0339 0.0255 21.084 0.478
MDA-MB-468 FIMM 10.815 N/A 0.237 73.395 0.0697
MFM-223 FIMM 54.913 0.0299 0.0184 19.016 0.502
SK-BR-3 FIMM 59.855 0.0192 0.0157 14.513 0.566
T47D FIMM 20.034 2.41 1.87 8.450 0.151
ZR-75-1 FIMM 40.831 6.99e-05 5.75e-05 27.109 0.383
CAL-148 FIMM 48.524 0.0681 0.0538 14.442 0.451
CAL-51 FIMM 35.585 0.363 0.344 3.104 0.323
CAL-85-1 FIMM 33.663 0.257 0.191 21.672 0.307
DU-4475 FIMM 59.590 0.0404 0.0403 0.468 0.586
HDQ-P1 FIMM 39.999 0.139 0.0869 22.362 0.359
MDA-MB-453 FIMM 64.440 0.0199 0.0189 5.356 0.623
KPL-1 CTRPv2 6.661 N/A 1e+06 52.550 0
CAL-120 CTRPv2 1.831 N/A 13.7 78.497 0.007
HDQ-P1 CTRPv2 33.218 0.761 0.208 31.876 0.278
JIMT-1 CTRPv2 26.970 2.16 0.27 41.741 0.216
HARA CTRPv2 34.878 0.546 0.321 21.761 0.308
CAMA-1 CTRPv2 23.386 N/A 0.00275 64.388 0.149
MCF7 CTRPv2 22.948 N/A 0.11 60.899 0.183
HCC1806 CTRPv2 33.347 0.202 0.129 41.558 0.299
HCC1954 CTRPv2 35.605 0.114 0.0664 44.305 0.317
HMC-1-8 CTRPv2 31.758 0.296 0.175 36.949 0.285
HCC1937 CTRPv2 23.817 N/A 0.231 50.104 0.183
HCC1395 CTRPv2 9.272 N/A 0.663 72.154 0.0608
CAL-51 CTRPv2 39.562 0.316 0.257 15.236 0.369
MDA-MB-231 CTRPv2 22.561 1.93 1.6 22.500 0.208
HCC1143 CTRPv2 31.966 0.58 0.292 29.643 0.281
ZR-75-1 CTRPv2 35.408 0.0885 0.0553 42.354 0.318
HCC1428 CTRPv2 21.960 N/A 0.00993 71.822 0.153
HCC38 CTRPv2 49.267 0.0798 0.0423 22.709 0.445
BT-549 CTRPv2 17.273 N/A 0.096 69.227 0.124
HCC202 CTRPv2 38.057 0.151 0.0168 47.694 0.323
DU-4475 CTRPv2 60.776 0.0573 0.0568 0.634 0.585
HCC1500 CTRPv2 43.642 0.263 0.041 29.618 0.374
Hs-578-T CTRPv2 43.033 1.1 1.1 0.000 0.367
MDA-MB-468 CTRPv2 15.573 3.19 1.5 47.551 0.133
CAL-85-1 CTRPv2 29.438 1.55 1.16 10.543 0.251
BT-20 CTRPv2 23.472 N/A 0.0652 60.193 0.16
UACC-812 CTRPv2 53.182 0.0123 0.00671 33.767 0.485
HCC1419 CTRPv2 12.252 N/A 0.111 77.600 0.0713
ZR-75-30 CTRPv2 25.506 N/A 0.113 53.255 0.216
MDA-MB-157 CTRPv2 32.422 0.511 0.443 21.744 0.306
MDA-MB-361 CTRPv2 90.680 1.84e-05 1.11e-05 7.902 0.896
T47D CTRPv2 16.200 N/A 1.06 51.034 0.123
BT-474 CTRPv2 29.129 N/A 0.0595 52.029 0.25
HCC2218 CTRPv2 35.939 0.109 0.0755 38.498 0.327
SK-BR-3 CTRPv2 39.791 0.191 0.0103 48.356 0.336
MDA-MB-453 CTRPv2 57.452 0.0225 0.0133 23.160 0.531
AU565 CTRPv2 38.650 0.423 0.015 46.978 0.321
MDA-MB-415 CTRPv2 52.227 0.0428 0.0195 26.333 0.473
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