| PLX4720 | CCLE, GDSC1000, CTRPv2 | 3192 |
| BMS-536924 | GDSC1000, CTRPv2 | 2234 |
| Sorafenib | CCLE, GDSC1000, GRAY, FIMM, CTRPv2 | 1939 |
| linifanib | GDSC1000, CTRPv2 | 1844 |
| foretinib | GDSC1000, CTRPv2 | 1825 |
| tivozanib | GDSC1000, CTRPv2 | 1822 |
| Axitinib | GDSC1000, FIMM, CTRPv2 | 1800 |
| OSI-930 | GDSC1000, CTRPv2 | 1680 |
| Vandetanib | CCLE, FIMM, CTRPv2 | 1381 |
| Sunitinib | GDSC1000, FIMM, CTRPv2 | 1319 |