| Erlotinib | CCLE, GDSC1000, gCSI, GRAY, FIMM, CTRPv2, UHNBreast | 2345 |
| lapatinib | CCLE, GDSC1000, gCSI, GRAY, FIMM, CTRPv2, UHNBreast | 2302 |
| BMS-536924 | GDSC1000, CTRPv2 | 2234 |
| Vandetanib | CCLE, FIMM, CTRPv2 | 1381 |
| CP724714 | GDSC1000 | 980 |
| CUDC-101 | GDSC1000 | 975 |
| neratinib | CTRPv2 | 867 |
| canertinib | CTRPv2 | 818 |
| WZ4002 | CTRPv2 | 614 |