| BMS-536924 | GDSC1000, CTRPv2 | 2234 |
| PHA-793887 | GDSC1000, CTRPv2 | 1848 |
| Bosutinib | GDSC1000, GRAY, FIMM, CTRPv2 | 1831 |
| BX-912 | GDSC1000 | 984 |
| AT-7519 | GDSC1000 | 984 |
| BX-795 | GDSC1000 | 889 |
| PF-573228 | CTRPv2 | 857 |
| SNS-032 | CTRPv2 | 795 |
| SB 216763 | GDSC1000 | 787 |
| Roscovitine | GDSC1000, FIMM | 472 |