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GSK429286A

Synonyms

SourcesNames Used
GDSC1000GSK429286A
PharmacoGx GSK429286A

External IDs

DatabaseIdentifier
Smiles: CC1=C(C(CC(=O)N1)c1ccc(cc1)C(F)(F)F)C(=O)Nc1cc2cn[nH]c2cc1F
Pubchem: 11373846

Annotated Targets

ROCK1

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK429286A


Feature TypeStandardized
Nominal ANOVA
mRNA IRF3 GDSC1000 pan-cancer AAC -0.088 0.01
mRNA HN1 GDSC1000 pan-cancer AAC 0.088 0.01
mRNA KRT8 GDSC1000 pan-cancer AAC -0.14 0.01
mRNA GPRASP2 GDSC1000 pan-cancer AAC 0.098 0.01
mRNA CDKN2C GDSC1000 pan-cancer AAC 0.09 0.01
mRNA RAD54B GDSC1000 pan-cancer AAC 0.084 0.01
mRNA TM9SF3 GDSC1000 pan-cancer AAC -0.085 0.01
mRNA RAB20 GDSC1000 pan-cancer AAC -0.092 0.01
mRNA ADGRG1 GDSC1000 pan-cancer AAC -0.098 0.01
mRNA AADACL2 GDSC1000 pan-cancer AAC 0.081 0.01
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