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GSK429286A

Synonyms

SourcesNames Used
GDSC1000GSK429286A
PharmacoGx GSK429286A

External IDs

DatabaseIdentifier
Smiles: CC1=C(C(CC(=O)N1)c1ccc(cc1)C(F)(F)F)C(=O)Nc1cc2cn[nH]c2cc1F
Pubchem: 11373846

Annotated Targets

ROCK1

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK429286A


Feature TypeStandardized
Nominal ANOVA
mRNA SKIL GDSC1000 pan-cancer AAC -0.093 0.006
mRNA SLC23A2 GDSC1000 pan-cancer AAC -0.098 0.006
mRNA TRIM24 GDSC1000 pan-cancer AAC 0.094 0.006
mRNA ATP6AP1L GDSC1000 pan-cancer AAC 0.088 0.006
mRNA XPO1 GDSC1000 pan-cancer AAC 0.089 0.006
mRNA OSBPL9 GDSC1000 pan-cancer AAC -0.091 0.006
mRNA CHEK1 GDSC1000 pan-cancer AAC 0.095 0.006
mRNA SLC44A3 GDSC1000 pan-cancer AAC -0.11 0.006
mRNA HLA-DRA GDSC1000 pan-cancer AAC -0.11 0.006
mRNA WDR5 GDSC1000 pan-cancer AAC 0.09 0.006
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