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GSK429286A

Synonyms

SourcesNames Used
GDSC1000GSK429286A
PharmacoGx GSK429286A

External IDs

DatabaseIdentifier
Smiles: CC1=C(C(CC(=O)N1)c1ccc(cc1)C(F)(F)F)C(=O)Nc1cc2cn[nH]c2cc1F
Pubchem: 11373846

Annotated Targets

ROCK1

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK429286A


Feature TypeStandardized
Nominal ANOVA
mRNA KLHL8 GDSC1000 pan-cancer AAC 0.11 0.005
mRNA CD8A GDSC1000 pan-cancer AAC 0.09 0.005
mRNA CLEC5A GDSC1000 pan-cancer AAC 0.09 0.005
mRNA OSBPL5 GDSC1000 pan-cancer AAC 0.092 0.005
mRNA CDC25A GDSC1000 pan-cancer AAC 0.11 0.005
mRNA SOCS2 GDSC1000 pan-cancer AAC 0.091 0.005
mRNA DHRS7 GDSC1000 pan-cancer AAC -0.096 0.005
mRNA TMEM156 GDSC1000 pan-cancer AAC -0.094 0.005
mRNA ZW10 GDSC1000 pan-cancer AAC 0.092 0.005
mRNA UXS1 GDSC1000 pan-cancer AAC -0.098 0.005
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