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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA IKZF1 GDSC1000 pan-cancer AAC 0.38 1e-07
mRNA ARHGAP30 GDSC1000 pan-cancer AAC 0.3 3e-06
mRNA P2RY8 GDSC1000 pan-cancer AAC 0.27 2e-06
mRNA CD53 GDSC1000 pan-cancer AAC 0.25 7e-05
mRNA ARHGAP15 GDSC1000 pan-cancer AAC 0.24 0.0003
mRNA LRMP GDSC1000 pan-cancer AAC 0.23 9e-07
mRNA ACAP1 GDSC1000 pan-cancer AAC 0.23 1e-05
mRNA PRPF4B GDSC1000 pan-cancer AAC 0.22 7e-13
mRNA CCAR1 GDSC1000 pan-cancer AAC 0.22 2e-11
mRNA CCDC88C GDSC1000 pan-cancer AAC 0.22 6e-09
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