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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA ABCB1 GDSC1000 pan-cancer AAC -0.29 6e-19
mRNA GNG12 GDSC1000 pan-cancer AAC -0.25 6e-09
mRNA NCKAP1 GDSC1000 pan-cancer AAC -0.23 4e-05
mRNA CD63 GDSC1000 pan-cancer AAC -0.22 1e-09
mRNA NQO1 GDSC1000 pan-cancer AAC -0.22 6e-09
mRNA TJP1 GDSC1000 pan-cancer AAC -0.22 0.0001
mRNA DUSP3 GDSC1000 pan-cancer AAC -0.21 1e-10
mRNA PPIC GDSC1000 pan-cancer AAC -0.21 1e-07
mRNA PRKD1 GDSC1000 pan-cancer AAC -0.21 2e-09
mRNA SHISA4 GDSC1000 pan-cancer AAC -0.21 9e-09
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