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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA C6orf203 GDSC1000 pan-cancer AAC 0.15 4e-07
mRNA TGOLN2 GDSC1000 pan-cancer AAC -0.16 4e-07
mRNA ZNF253 GDSC1000 pan-cancer AAC 0.16 5e-07
mRNA SLTM GDSC1000 pan-cancer AAC 0.16 5e-07
mRNA PMP22 GDSC1000 pan-cancer AAC -0.18 5e-07
mRNA AVPI1 GDSC1000 pan-cancer AAC -0.18 5e-07
mRNA CNRIP1 GDSC1000 pan-cancer AAC -0.2 6e-07
mRNA ANKRD46 GDSC1000 pan-cancer AAC 0.16 6e-07
mRNA MAP3K4 GDSC1000 pan-cancer AAC 0.16 6e-07
mRNA UBE3D GDSC1000 pan-cancer AAC 0.16 6e-07
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