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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA SPINT1 GDSC1000 pan-cancer AAC 0.13 0.0007
mRNA RNPC3 GDSC1000 pan-cancer AAC 0.11 0.0007
mRNA INPP5F GDSC1000 pan-cancer AAC -0.12 0.0007
mRNA WSB2 GDSC1000 pan-cancer AAC -0.12 0.0007
mRNA ZNF554 GDSC1000 pan-cancer AAC 0.098 0.0007
mRNA PER2 GDSC1000 pan-cancer AAC 0.11 0.0007
mRNA TNFRSF1A GDSC1000 pan-cancer AAC -0.11 0.0007
mRNA SLA GDSC1000 pan-cancer AAC 0.12 0.0007
mRNA FBXW7 GDSC1000 pan-cancer AAC 0.11 0.0007
mRNA ATP8B2 GDSC1000 pan-cancer AAC -0.11 0.0007
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