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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA C1orf35 GDSC1000 pan-cancer AAC 0.089 0.004
mRNA SCARA3 GDSC1000 pan-cancer AAC -0.091 0.004
mRNA MED15 GDSC1000 pan-cancer AAC -0.087 0.004
mRNA TET2 GDSC1000 pan-cancer AAC 0.087 0.004
mRNA RAB11FIP5 GDSC1000 pan-cancer AAC -0.11 0.004
mRNA RILP GDSC1000 pan-cancer AAC -0.086 0.004
mRNA GPR87 GDSC1000 pan-cancer AAC 0.11 0.004
mRNA GPR153 GDSC1000 pan-cancer AAC 0.085 0.004
mRNA NFX1 GDSC1000 pan-cancer AAC 0.096 0.004
mRNA PCDHB3 GDSC1000 pan-cancer AAC -0.082 0.004
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