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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA CHD7 GDSC1000 pan-cancer AAC 0.096 0.003
mRNA KDM1A GDSC1000 pan-cancer AAC 0.089 0.003
mRNA EMSY GDSC1000 pan-cancer AAC 0.089 0.003
mRNA UNC5B GDSC1000 pan-cancer AAC 0.097 0.003
mRNA EIF4H GDSC1000 pan-cancer AAC 0.084 0.003
mRNA CPNE8 GDSC1000 pan-cancer AAC -0.091 0.003
mRNA LRRC59 GDSC1000 pan-cancer AAC -0.086 0.003
mRNA ABLIM3 GDSC1000 pan-cancer AAC -0.096 0.003
mRNA DYNLRB1 GDSC1000 pan-cancer AAC -0.09 0.003
mRNA XRCC5 GDSC1000 pan-cancer AAC 0.091 0.003
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