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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA TBPL1 GDSC1000 pan-cancer AAC 0.092 0.003
mRNA HDAC1 GDSC1000 pan-cancer AAC 0.094 0.003
mRNA INTS6 GDSC1000 pan-cancer AAC 0.09 0.003
mRNA ZAP70 GDSC1000 pan-cancer AAC 0.096 0.003
mRNA MT2A GDSC1000 pan-cancer AAC -0.1 0.003
mRNA FASTK GDSC1000 pan-cancer AAC -0.091 0.003
mRNA PIK3R5 GDSC1000 pan-cancer AAC 0.098 0.003
mRNA DIO2 GDSC1000 pan-cancer AAC -0.092 0.003
mRNA TENM3 GDSC1000 pan-cancer AAC -0.099 0.003
mRNA UBA5 GDSC1000 pan-cancer AAC 0.091 0.003
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