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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA POLE4 GDSC1000 pan-cancer AAC -0.091 0.002
mRNA CEP192 GDSC1000 pan-cancer AAC 0.092 0.002
mRNA MRS2 GDSC1000 pan-cancer AAC 0.091 0.002
mRNA IFNGR1 GDSC1000 pan-cancer AAC 0.092 0.002
mRNA KCNAB1 GDSC1000 pan-cancer AAC -0.096 0.002
mRNA DCT GDSC1000 pan-cancer AAC -0.12 0.002
mRNA RIC1 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA PPA1 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA SERPINC1 GDSC1000 pan-cancer AAC -0.093 0.002
mRNA ANKRD33 GDSC1000 pan-cancer AAC 0.089 0.002
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