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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA MTO1 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA RNF220 GDSC1000 pan-cancer AAC 0.093 0.002
mRNA TGFB1I1 GDSC1000 pan-cancer AAC -0.11 0.002
mRNA DPY19L1 GDSC1000 pan-cancer AAC -0.096 0.002
mRNA HMGN3 GDSC1000 pan-cancer AAC 0.092 0.002
mRNA RFX3 GDSC1000 pan-cancer AAC 0.096 0.002
mRNA SNX21 GDSC1000 pan-cancer AAC -0.098 0.002
mRNA PDK4 GDSC1000 pan-cancer AAC -0.092 0.002
mRNA OR1M1 GDSC1000 pan-cancer AAC 0.091 0.002
mRNA ALG9 GDSC1000 pan-cancer AAC 0.093 0.002
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