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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA SLC35C2 GDSC1000 pan-cancer AAC -0.093 0.002
mRNA STOML2 GDSC1000 pan-cancer AAC 0.09 0.002
mRNA POLR2G GDSC1000 pan-cancer AAC 0.092 0.002
mRNA ATAD2 GDSC1000 pan-cancer AAC 0.095 0.002
mRNA ZNF84 GDSC1000 pan-cancer AAC 0.095 0.002
mRNA C1orf52 GDSC1000 pan-cancer AAC 0.089 0.002
mRNA TIMP3 GDSC1000 pan-cancer AAC -0.11 0.002
mRNA MTERF3 GDSC1000 pan-cancer AAC 0.093 0.002
mRNA PARD6G GDSC1000 pan-cancer AAC 0.1 0.002
mRNA ARHGAP1 GDSC1000 pan-cancer AAC -0.096 0.002
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