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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA RABEP1 GDSC1000 pan-cancer AAC 0.094 0.001
mRNA ZNF558 GDSC1000 pan-cancer AAC 0.093 0.002
mRNA ZBTB39 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA ZNF431 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA C16orf87 GDSC1000 pan-cancer AAC 0.1 0.002
mRNA USP42 GDSC1000 pan-cancer AAC 0.094 0.002
mRNA PRUNE1 GDSC1000 pan-cancer AAC 0.096 0.002
mRNA TMEM192 GDSC1000 pan-cancer AAC -0.095 0.002
mRNA ARHGEF4 GDSC1000 pan-cancer AAC 0.099 0.002
mRNA CXCL2 GDSC1000 pan-cancer AAC -0.1 0.002
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