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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA MMS22L GDSC1000 pan-cancer AAC 0.098 0.001
mRNA MBD3 GDSC1000 pan-cancer AAC 0.097 0.001
mRNA CLCA2 GDSC1000 pan-cancer AAC 0.099 0.001
mRNA LAPTM5 GDSC1000 pan-cancer AAC 0.16 0.001
mRNA PHF3 GDSC1000 pan-cancer AAC 0.099 0.001
mRNA SH3YL1 GDSC1000 pan-cancer AAC 0.11 0.001
mRNA DAAM2 GDSC1000 pan-cancer AAC -0.12 0.001
mRNA FAM177A1 GDSC1000 pan-cancer AAC -0.12 0.001
mRNA SEPT1 GDSC1000 pan-cancer AAC 0.12 0.001
mRNA HNRNPF GDSC1000 pan-cancer AAC 0.1 0.001
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