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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA ZBTB44 GDSC1000 pan-cancer AAC 0.1 0.001
mRNA PRKAG1 GDSC1000 pan-cancer AAC -0.1 0.001
mRNA HIST1H3F GDSC1000 pan-cancer AAC 0.1 0.001
mRNA MARK2 GDSC1000 pan-cancer AAC 0.1 0.001
mRNA PRR16 GDSC1000 pan-cancer AAC -0.1 0.001
mRNA NBL1 GDSC1000 pan-cancer AAC -0.12 0.001
mRNA FARP1 GDSC1000 pan-cancer AAC -0.12 0.001
mRNA GPX8 GDSC1000 pan-cancer AAC -0.13 0.001
mRNA DUSP19 GDSC1000 pan-cancer AAC -0.097 0.001
mRNA MAP2K7 GDSC1000 pan-cancer AAC 0.098 0.001
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