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AT-7519

Synonyms

SourcesNames Used
GDSC1000AT-7519
PharmacoGx AT-7519

External IDs

DatabaseIdentifier
Smiles: Clc1cccc(Cl)c1C(=O)Nc1c[nH]nc1C(=O)NC1CCNCC1
Pubchem: 11338033

Annotated Targets

CDK14, CDK1, CDK2, CDK4, CDK5, CDK6, CDK9

FDA Approval Status

Not Approved
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Top molecular features associated with response to AT-7519


Feature TypeStandardized
Nominal ANOVA
mRNA ABRACL GDSC1000 pan-cancer AAC 0.088 0.004
mRNA ATG2B GDSC1000 pan-cancer AAC 0.087 0.004
mRNA POLR3F GDSC1000 pan-cancer AAC 0.083 0.004
mRNA F2 GDSC1000 pan-cancer AAC -0.089 0.004
mRNA PTPRE GDSC1000 pan-cancer AAC 0.089 0.004
mRNA ZNF197 GDSC1000 pan-cancer AAC 0.087 0.004
mRNA PKN2 GDSC1000 pan-cancer AAC 0.094 0.004
mRNA ZNF510 GDSC1000 pan-cancer AAC 0.084 0.004
mRNA EFS GDSC1000 pan-cancer AAC 0.09 0.004
mRNA UPF1 GDSC1000 pan-cancer AAC 0.088 0.004
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