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barasertib

Synonyms

SourcesNames Used
CTRPv2barasertib
PharmacoGx barasertib

External IDs

DatabaseIdentifier
Smiles: CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)[nH]n3)ncnc2c1
Pubchem: 11497983

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to barasertib


Feature TypeStandardized
Nominal ANOVA
mRNA EHMT2 CTRPv2 pan-cancer AAC 0.28 4e-16
mRNA ILF3 CTRPv2 pan-cancer AAC 0.28 7e-16
mRNA ZNF445 CTRPv2 pan-cancer AAC 0.29 7e-16
mRNA SPNS3 CTRPv2 pan-cancer AAC 0.27 7e-16
mRNA GRK2 CTRPv2 pan-cancer AAC 0.33 9e-16
mRNA SUGP2 CTRPv2 pan-cancer AAC 0.3 3e-15
mRNA SOX4 CTRPv2 pan-cancer AAC 0.25 4e-15
mRNA HNRNPA0 CTRPv2 pan-cancer AAC 0.26 5e-15
mRNA DOT1L CTRPv2 pan-cancer AAC 0.31 5e-15
mRNA SCAF4 CTRPv2 pan-cancer AAC 0.29 6e-15
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