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alisertib

Synonyms

SourcesNames Used
CTRPv2alisertib
PharmacoGx alisertib

External IDs

DatabaseIdentifier
Smiles: COc1cc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2OC)ccc1C(O)=O
Pubchem: 24771867

Annotated Targets

AURKA, AURKB

FDA Approval Status

Not Approved
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Top molecular features associated with response to alisertib


Feature TypeStandardized
Nominal ANOVA
mRNA HNRNPA1 CTRPv2 pan-cancer AAC 0.32 6e-19
mRNA CBX2 CTRPv2 pan-cancer AAC 0.3 1e-18
mRNA MBTD1 CTRPv2 pan-cancer AAC 0.3 9e-16
mRNA ZBED4 CTRPv2 pan-cancer AAC 0.29 9e-16
mRNA KHDRBS1 CTRPv2 pan-cancer AAC 0.26 7e-15
mRNA MEX3A CTRPv2 pan-cancer AAC 0.3 8e-15
mRNA LMNB1 CTRPv2 pan-cancer AAC 0.26 3e-14
mRNA ARHGAP19 CTRPv2 pan-cancer AAC 0.29 4e-14
mRNA ARHGAP19-SLIT1 CTRPv2 pan-cancer AAC 0.28 1e-13
mRNA FAM117B CTRPv2 pan-cancer AAC 0.24 1e-13
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