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regorafenib

Synonyms

SourcesNames Used
CTRPv2regorafenib
PharmacoGx regorafenib

External IDs

DatabaseIdentifier
Pubchem: 11167602

Annotated Targets

FRK, DDR2, MAPK11, KIT, BRAF, TEK, ABL1, EPHA2, FGFR1, FGFR2, FLT1, FLT4, KDR, NTRK1, PDGFRA, PDGFRB, RAF1, RET

FDA Approval Status

Approved
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Top molecular features associated with response to regorafenib


Feature TypeStandardized
Nominal ANOVA
mRNA EPX CTRPv2 pan-cancer AAC 0.24 2e-11
mRNA TOP1MT CTRPv2 pan-cancer AAC 0.26 4e-11
mRNA HRH4 CTRPv2 pan-cancer AAC 0.24 4e-11
mRNA CCR6 CTRPv2 pan-cancer AAC 0.24 5e-11
mRNA KCNN2 CTRPv2 pan-cancer AAC 0.25 1e-10
mRNA PPP1R27 CTRPv2 pan-cancer AAC 0.23 1e-10
mRNA IL3RA CTRPv2 pan-cancer AAC 0.25 1e-10
mRNA SENP6 CTRPv2 pan-cancer AAC 0.24 2e-10
mRNA MS4A6A CTRPv2 pan-cancer AAC 0.23 2e-10
mRNA PIM1 CTRPv2 pan-cancer AAC 0.24 3e-10
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