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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA ZXDC GDSC1000 pan-cancer AAC -0.063 0.07
mRNA ZSWIM5 GDSC1000 pan-cancer AAC -0.067 0.07
mRNA ZSCAN18 GDSC1000 pan-cancer AAC -0.076 0.04
mRNA ZPBP2 GDSC1000 pan-cancer AAC 0.12 0.0003
mRNA ZP4 GDSC1000 pan-cancer AAC 0.076 0.02
mRNA ZNF99 GDSC1000 pan-cancer AAC -0.063 0.07
mRNA ZNF883 GDSC1000 pan-cancer AAC -0.063 0.08
mRNA ZNF880 GDSC1000 pan-cancer AAC -0.098 0.007
mRNA ZNF853 GDSC1000 pan-cancer AAC -0.064 0.08
mRNA ZNF844 GDSC1000 pan-cancer AAC -0.11 0.002
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