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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA SPCS1 GDSC1000 pan-cancer AAC -0.093 0.01
mRNA ECM2 GDSC1000 pan-cancer AAC 0.092 0.01
mRNA PPP1R1C GDSC1000 pan-cancer AAC 0.088 0.01
mRNA PTGS2 GDSC1000 pan-cancer AAC 0.093 0.01
mRNA MSX1 GDSC1000 pan-cancer AAC -0.089 0.01
mRNA LPAR5 GDSC1000 pan-cancer AAC 0.098 0.01
mRNA C9orf43 GDSC1000 pan-cancer AAC -0.087 0.01
mRNA PPP1R13L GDSC1000 pan-cancer AAC 0.11 0.01
mRNA DYNLRB1 GDSC1000 pan-cancer AAC -0.091 0.01
mRNA C3 GDSC1000 pan-cancer AAC 0.097 0.01
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