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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA TACC1 GDSC1000 pan-cancer AAC -0.073 0.05
mRNA AHNAK2 GDSC1000 pan-cancer AAC 0.08 0.05
mRNA MRS2 GDSC1000 pan-cancer AAC -0.066 0.05
mRNA EZR GDSC1000 pan-cancer AAC 0.074 0.05
mRNA MUC12 GDSC1000 pan-cancer AAC -0.068 0.05
mRNA KCNN4 GDSC1000 pan-cancer AAC 0.068 0.05
mRNA SLC44A5 GDSC1000 pan-cancer AAC 0.069 0.05
mRNA PRR27 GDSC1000 pan-cancer AAC 0.065 0.05
mRNA AP4E1 GDSC1000 pan-cancer AAC 0.071 0.05
mRNA DSG3 GDSC1000 pan-cancer AAC 0.087 0.05
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