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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA NDUFB11 GDSC1000 pan-cancer AAC -0.071 0.05
mRNA VN1R4 GDSC1000 pan-cancer AAC 0.069 0.05
mRNA ARSJ GDSC1000 pan-cancer AAC 0.077 0.05
mRNA PPFIA3 GDSC1000 pan-cancer AAC -0.073 0.05
mRNA ARHGAP42 GDSC1000 pan-cancer AAC 0.07 0.05
mRNA ACVR2B GDSC1000 pan-cancer AAC -0.072 0.05
mRNA IP6K1 GDSC1000 pan-cancer AAC -0.074 0.05
mRNA RPGRIP1L GDSC1000 pan-cancer AAC 0.07 0.05
mRNA GNG7 GDSC1000 pan-cancer AAC -0.084 0.05
mRNA CDKN1C GDSC1000 pan-cancer AAC -0.068 0.05
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