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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA OSBPL10 GDSC1000 pan-cancer AAC 0.073 0.04
mRNA PRELID3B GDSC1000 pan-cancer AAC -0.073 0.04
mRNA FRA10AC1 GDSC1000 pan-cancer AAC 0.069 0.04
mRNA FBXL19 GDSC1000 pan-cancer AAC 0.071 0.04
mRNA ANLN GDSC1000 pan-cancer AAC 0.075 0.04
mRNA LPIN2 GDSC1000 pan-cancer AAC -0.072 0.04
mRNA GLT8D2 GDSC1000 pan-cancer AAC 0.08 0.04
mRNA PLEKHA4 GDSC1000 pan-cancer AAC -0.077 0.04
mRNA HTT GDSC1000 pan-cancer AAC -0.07 0.04
mRNA CPQ GDSC1000 pan-cancer AAC -0.079 0.04
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