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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA PRR25 GDSC1000 pan-cancer AAC -0.065 0.06
mRNA ISCU GDSC1000 pan-cancer AAC -0.067 0.06
mRNA FGFR4 GDSC1000 pan-cancer AAC -0.072 0.06
mRNA CHCHD3 GDSC1000 pan-cancer AAC -0.066 0.06
mRNA HRH1 GDSC1000 pan-cancer AAC 0.073 0.06
mRNA CAMTA2 GDSC1000 pan-cancer AAC -0.064 0.06
mRNA UBE2O GDSC1000 pan-cancer AAC -0.069 0.06
mRNA ARSI GDSC1000 pan-cancer AAC 0.07 0.06
mRNA ZNF66 GDSC1000 pan-cancer AAC 0.063 0.06
mRNA GPR83 GDSC1000 pan-cancer AAC -0.065 0.06
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