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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA ATF7IP2 GDSC1000 pan-cancer AAC 0.071 0.06
mRNA AMMECR1 GDSC1000 pan-cancer AAC 0.066 0.06
mRNA ARHGAP18 GDSC1000 pan-cancer AAC 0.07 0.06
mRNA NKX3-2 GDSC1000 pan-cancer AAC -0.068 0.06
mRNA TMEM134 GDSC1000 pan-cancer AAC -0.072 0.06
mRNA DIMT1 GDSC1000 pan-cancer AAC 0.068 0.06
mRNA LPIN3 GDSC1000 pan-cancer AAC -0.079 0.06
mRNA OR1A1 GDSC1000 pan-cancer AAC 0.066 0.06
mRNA SND1 GDSC1000 pan-cancer AAC -0.07 0.06
mRNA DNAJC27 GDSC1000 pan-cancer AAC -0.068 0.06
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