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XAV-939

Synonyms

SourcesNames Used
GDSC1000XAV939
PharmacoGx XAV-939

External IDs

DatabaseIdentifier
Smiles: C1CSCC2=C1NC(=NC2=O)C3=CC=C(C=C3)C(F)(F)F
Inchikey: KLGQSVMIPOVQAX-UHFFFAOYSA-N
Pubchem: 2726824

Annotated Targets

TNKS, TNKS2

FDA Approval Status

Not Approved
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Top molecular features associated with response to XAV-939


Feature TypeStandardized
Nominal ANOVA
mRNA EXD3 GDSC1000 pan-cancer AAC -0.069 0.05
mRNA BIRC2 GDSC1000 pan-cancer AAC 0.069 0.05
mRNA LPAR6 GDSC1000 pan-cancer AAC 0.071 0.05
mRNA AVPR1B GDSC1000 pan-cancer AAC -0.067 0.05
mRNA TRPC3 GDSC1000 pan-cancer AAC -0.067 0.05
mRNA PSMA3 GDSC1000 pan-cancer AAC 0.07 0.05
mRNA ROM1 GDSC1000 pan-cancer AAC -0.07 0.05
mRNA TMEM123 GDSC1000 pan-cancer AAC 0.071 0.05
mRNA LOX GDSC1000 pan-cancer AAC 0.079 0.05
mRNA IGSF8 GDSC1000 pan-cancer AAC -0.076 0.05
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