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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA PPP2R3B CTRPv2 pan-cancer AAC 0.19 5e-05
mRNA BCL7A CTRPv2 pan-cancer AAC 0.19 0.0001
mRNA C19orf47 CTRPv2 pan-cancer AAC 0.19 3e-05
mRNA DBNL CTRPv2 pan-cancer AAC 0.2 2e-05
mRNA LDAH CTRPv2 pan-cancer AAC 0.2 0.0001
mRNA GGA2 CTRPv2 pan-cancer AAC 0.2 0.0001
mRNA PTOV1 CTRPv2 pan-cancer AAC 0.2 1e-05
mRNA FBXO10 CTRPv2 pan-cancer AAC 0.2 3e-05
mRNA PRR3 CTRPv2 pan-cancer AAC 0.21 0.0001
mRNA MEX3C CTRPv2 pan-cancer AAC 0.21 3e-05
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