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Crizotinib

Synonyms

SourcesNames Used
CCLE, GRAYPF-2341066
GDSC1000, FIMMCrizotinib
gCSI, CTRPv2crizotinib
PharmacoGx Crizotinib

External IDs

DatabaseIdentifier
Smiles: CC(C1=C(C=C(C=C1Cl)F)Cl)OC2=C(N=CC(=C2)C3=CN(N=C3)C4CCNCC4)N
Inchikey: SCJHEFQWKWHQTO-GFCCVEGCSA-N
Pubchem: 54613769

Annotated Targets

MET, ALK

FDA Approval Status

Approved
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Top molecular features associated with response to Crizotinib


Feature TypeStandardized
Nominal ANOVA
mRNA CPTP FIMM pan-cancer AAC -0.58 0.0009
mRNA CPSF3L FIMM pan-cancer AAC -0.52 0.001
mRNA ZBTB7B FIMM pan-cancer AAC -0.52 0.003
mRNA SLC30A1 FIMM pan-cancer AAC -0.5 0.002
mRNA KRT37 FIMM pan-cancer AAC -0.5 0.003
mRNA LRMP GDSC1000 pan-cancer AAC -0.43 5e-07
mRNA MAP4K1 gCSI pan-cancer AAC -0.42 3e-05
mRNA EAF2 GDSC1000 pan-cancer AAC -0.4 2e-07
mRNA RCSD1 gCSI pan-cancer AAC -0.39 0.0009
mRNA LRMP gCSI pan-cancer AAC -0.35 0.0002
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