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Crizotinib

Synonyms

SourcesNames Used
CCLE, GRAYPF-2341066
GDSC1000, FIMMCrizotinib
gCSI, CTRPv2crizotinib
PharmacoGx Crizotinib

External IDs

DatabaseIdentifier
Smiles: CC(C1=C(C=C(C=C1Cl)F)Cl)OC2=C(N=CC(=C2)C3=CN(N=C3)C4CCNCC4)N
Inchikey: SCJHEFQWKWHQTO-GFCCVEGCSA-N
Pubchem: 54613769

Annotated Targets

MET, ALK

FDA Approval Status

Approved
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Top molecular features associated with response to Crizotinib


Feature TypeStandardized
Nominal ANOVA
mRNA CCDC125 GDSC1000 pan-cancer AAC 0.31 3e-09
mRNA HAVCR2 GDSC1000 pan-cancer AAC 0.32 4e-09
mRNA PGC CTRPv2 pan-cancer AAC 0.18 4e-09
mRNA FAM129B GDSC1000 pan-cancer AAC 0.47 4e-09
mRNA TMPRSS11F CTRPv2 pan-cancer AAC 0.18 5e-09
mRNA ATP6V0A4 CTRPv2 pan-cancer AAC 0.19 7e-09
mRNA HGF CCLE pan-cancer AAC 0.27 7e-09
mRNA PTPN7 CTRPv2 pan-cancer AAC 0.26 7e-09
mRNA IL2RA GDSC1000 pan-cancer AAC 0.3 8e-09
mRNA MTMR7 GDSC1000 pan-cancer AAC 0.31 8e-09
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