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Crizotinib

Synonyms

SourcesNames Used
CCLE, GRAYPF-2341066
GDSC1000, FIMMCrizotinib
gCSI, CTRPv2crizotinib
PharmacoGx Crizotinib

External IDs

DatabaseIdentifier
Smiles: CC(C1=C(C=C(C=C1Cl)F)Cl)OC2=C(N=CC(=C2)C3=CN(N=C3)C4CCNCC4)N
Inchikey: SCJHEFQWKWHQTO-GFCCVEGCSA-N
Pubchem: 54613769

Annotated Targets

MET, ALK

FDA Approval Status

Approved
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Top molecular features associated with response to Crizotinib


Feature TypeStandardized
Nominal ANOVA
mRNA C14orf105 FIMM pan-cancer AAC 0.53 0.002
mRNA HNRNPH1 FIMM pan-cancer AAC 0.54 0.001
mRNA ALK GDSC1000 pan-cancer AAC 0.54 2e-28
mRNA PFDN4 FIMM pan-cancer AAC 0.55 0.0008
mRNA TDRD1 FIMM pan-cancer AAC 0.55 0.001
mRNA PPP1R12A FIMM pan-cancer AAC 0.56 0.002
mRNA KIAA1033 FIMM pan-cancer AAC 0.56 0.002
mRNA SPTLC1 FIMM pan-cancer AAC 0.57 0.001
mRNA MLLT10 FIMM pan-cancer AAC 0.57 0.001
mRNA TRMO FIMM pan-cancer AAC 0.57 0.0006
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