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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA L3MBTL2 CTRPv2 pan-cancer AAC 0.17 8e-06
mRNA ROGDI CTRPv2 pan-cancer AAC 0.17 8e-06
mRNA NLRP7 CTRPv2 pan-cancer AAC 0.16 8e-06
mRNA E2F2 CTRPv2 pan-cancer AAC 0.19 9e-06
mRNA SMIM14 CTRPv2 pan-cancer AAC 0.16 9e-06
mRNA ARHGAP45 CTRPv2 pan-cancer AAC 0.23 9e-06
mRNA P2RY8 CTRPv2 pan-cancer AAC 0.21 1e-05
mRNA NCF1 CTRPv2 pan-cancer AAC 0.17 1e-05
mRNA GTF2I CTRPv2 pan-cancer AAC 0.16 1e-05
mRNA RP11-212D19.4 CTRPv2 pan-cancer AAC -0.16 1e-05
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