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PLX4720

Synonyms

SourcesNames Used
CCLE, GDSC1000PLX4720
CTRPv2PLX-4720
PharmacoGx PLX4720

External IDs

DatabaseIdentifier
Smiles: CCCS(=O)(=O)NC1=C(C(=C(C=C1)F)C(=O)C2=CNC3=NC=C(C=C23)Cl)F
Inchikey: YZDJQTHVDDOVHR-UHFFFAOYSA-N
Pubchem: 24180719

Annotated Targets

BRAF, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to PLX4720


Feature TypeStandardized
Nominal ANOVA
mRNA A2M GDSC1000 pan-cancer AAC 0.16 4e-06
mRNA A4GNT GDSC1000 pan-cancer AAC -0.092 0.002
mRNA AARS2 CTRPv2 pan-cancer AAC 0.12 0.002
mRNA AASS GDSC1000 pan-cancer AAC 0.13 0.0001
mRNA ABC13-47488600E17.1 CTRPv2 pan-cancer AAC 0.1 0.003
mRNA ABCB4 CTRPv2 pan-cancer AAC 0.16 2e-05
mRNA ABCB5 CCLE pan-cancer AAC 0.2 1e-05
mRNA ABCD1 CTRPv2 pan-cancer AAC 0.13 0.0005
mRNA ABCG5 CCLE pan-cancer AAC 0.17 0.0001
mRNA ABHD17C CCLE pan-cancer AAC 0.16 0.002
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